| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CTSD |
US10889581, Example 112 |
NA |
176000 |
NA |
NA |
NA |
NA |
BindingDB |
| CTSD |
US10889581, Example 106 |
NA |
614300 |
NA |
NA |
NA |
NA |
BindingDB |
| CTSD |
US11021493, Example 277 |
NA |
213500 |
NA |
NA |
NA |
NA |
BindingDB |
| CTSD |
US11021493, Example 240 |
NA |
375400 |
NA |
NA |
NA |
NA |
BindingDB |
| CTSD |
US11021493, Example 261 |
NA |
178000 |
NA |
NA |
NA |
NA |
BindingDB |
| CTSD |
(1S,5S,6S)-3-amino-5-[5-[(5-chloropyridine-2-carbonyl)amino]-2,3-difluorophenyl]-N,5-dimethyl-2-thia-4-azabicyclo[4.1.0]hept-3-ene-1-carboxamide |
NA |
795000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSD |
[3-[3-(4-aminophenyl)-3-oxopropyl]-2,3,4,7-tetrahydro-1H-azepin-5-yl]methyl naphthalene-2-carboxylate |
NA |
262000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSD |
(2S)-2-[[(3S,4S)-3-hydroxy-6-methyl-4-(3-methylbutanoylamino)heptanoyl]amino]propanoic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CTSD |
US11021493, Example 101 |
NA |
211800 |
NA |
NA |
NA |
NA |
BindingDB |
| CTSD |
US11021493, Example 108 |
NA |
144600 |
NA |
NA |
NA |
NA |
BindingDB |
| CTSD |
US11021493, Example 219 |
NA |
208000 |
NA |
NA |
NA |
NA |
BindingDB |
| CTSD |
1,3-di(9H-carbazol-9-yl)propan-2-ol |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| CTSD |
Nafamostat |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| CTSD |
N-[3-[(4aR,7aS)-2-amino-4a,5,6,7-tetrahydro-4H-cyclopenta[d][1,3]thiazin-7a-yl]-4-fluorophenyl]-5-fluoropyridine-2-carboxamide |
NA |
3000000 |
NA |
NA |
NA |
NA |
TTD |
| CTSD |
2-Benzyl-N-[1-(1-cyclohexylmethyl-2,3,4,5,6-pentahydroxy-hexylcarbamoyl)-2-(1H-imidazol-4-yl)-ethyl]-3-(2-methyl-propane-2-sulfonyl)-propionamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CTSD |
2-[1-(3,4,5-Trimethoxybenzoyl)naphthalene-2-yloxy]-ethylethanoate |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CTSD |
4-(1-(3,4,5-Trimethoxybenzoyl)naphthalen-2-yloxy)but-2-enoic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CTSD |
N-phenyl-2-(1-(3,4,5-trimethoxybenzoyl)naphthalen-2-yloxy)acetamide |
NA |
231500 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSD |
N-phenyl-4-(1-(3,4,5-trimethoxybenzoyl)naphthalen-2-yloxy)but-2-enamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CTSD |
N-(4-methoxyphenyl)-2-(1-(3,4,5-trimethoxybenzoyl)naphthalen-2-yloxy)acetamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |