| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CTSD |
US9611261, Example 330 |
NA |
139000 |
NA |
NA |
NA |
NA |
BindingDB |
| CTSD |
US9611261, Example 419 |
NA |
275500 |
NA |
NA |
NA |
NA |
BindingDB |
| CTSD |
US10246429, Example 166 |
NA |
146500 |
NA |
NA |
NA |
NA |
BindingDB |
| CTSD |
US11021493, Example 184 |
NA |
335200 |
NA |
NA |
NA |
NA |
BindingDB |
| CTSD |
(4aR,7aR)-7a-[(1R,2R)-2-(2-{[(1R,2R)-2-methylcyclopropyl]methoxy}propan-2-yl)cyclopropyl]-6-(pyrimidin-2-yl)-4,4a,5,6,7,7a-hexahydropyrrolo[3,4-d][1,3]thiazin-2-amine |
NA |
160000 |
NA |
NA |
NA |
NA |
BindingDB |
| CTSD |
US10246429, Example 362 |
NA |
348510 |
NA |
NA |
NA |
NA |
BindingDB |
| CTSD |
N-[3-[(3R,6S)-5-amino-3,6-dimethyl-6-(trifluoromethyl)-2H-1,4-oxazin-3-yl]phenyl]-5-bromopyridine-2-carboxamide |
NA |
139000 |
NA |
NA |
NA |
NA |
BindingDB |
| CTSD |
N-[(4S)-2-amino-3'-cyclopropylspiro[5H-1,3-oxazole-4,5'-chromeno[2,3-c]pyridine]-7'-yl]-5-chloropyridine-2-carboxamide |
NA |
310000 |
NA |
NA |
NA |
NA |
TTD |
| CTSD |
N-[(4S)-2-amino-3'-methylspiro[5H-1,3-oxazole-4,5'-chromeno[2,3-c]pyridine]-7'-yl]-5-chloropyridine-2-carboxamide |
NA |
640000 |
NA |
NA |
NA |
NA |
TTD |
| CTSD |
N-[(4S)-2-amino-3'-chlorospiro[5H-1,3-oxazole-4,5'-chromeno[2,3-c]pyridine]-7'-yl]-5-chloropyridine-2-carboxamide |
NA |
1100000 |
NA |
NA |
NA |
NA |
TTD |
| CTSD |
N-[(4S)-2-amino-3'-methoxyspiro[5H-1,3-oxazole-4,5'-chromeno[2,3-c]pyridine]-7'-yl]-5-chloropyridine-2-carboxamide |
NA |
1200000 |
NA |
NA |
NA |
NA |
TTD |
| CTSD |
N-[(4S)-2-amino-3'-(oxan-4-yl)spiro[5H-1,3-oxazole-4,5'-chromeno[2,3-c]pyridine]-7'-yl]-5-chloropyridine-2-carboxamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| CTSD |
US10889581, Example 102 |
NA |
673000 |
NA |
NA |
NA |
NA |
BindingDB |
| CTSD |
US10889581, Example 105 |
NA |
500100 |
NA |
NA |
NA |
NA |
BindingDB |
| CTSD |
US10889581, Example 138 |
NA |
903300 |
NA |
NA |
NA |
NA |
BindingDB |
| CTSD |
US10889581, Example 108 |
NA |
783700 |
NA |
NA |
NA |
NA |
BindingDB |
| CTSD |
US10889581, Example 100 |
NA |
4866200 |
NA |
NA |
NA |
NA |
BindingDB |
| CTSD |
US10889581, Example 131 |
NA |
994800 |
NA |
NA |
NA |
NA |
BindingDB |
| CTSD |
US10889581, Example 126 |
NA |
268000 |
NA |
NA |
NA |
NA |
BindingDB |
| CTSD |
US10889581, Example 117 |
NA |
169000 |
NA |
NA |
NA |
NA |
BindingDB |