| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CTSL |
2-((S)-2-{(S)-3-Methoxy-2-[(pyrazine-2-carbonyl)-amino]-butyrylamino}-3,3-dimethyl-butyryl)-octahydro-cyclopenta[c]pyrrole-1-carboxylic acid (1-cyclopropylaminooxalyl-butyl)-amide |
146000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSL |
(5-Methylimidazo[1,2-a]pyridin-2-yl)methyl (pyridin-3-ylmethyl)carbamodithioate |
NA |
122000 |
NA |
NA |
NA |
NA |
BindingDB |
| CTSS |
(1r)-1-{[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]methyl}-2,2-dimethylpropyl(1S)-1-[oxo(1h-pyrazol-5-ylamino)acetyl]pentylcarbamate |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSS |
N-[(2S)-1-[[(1S)-1-cyano-2,2-dimethylpropyl]amino]-4-methyl-1-oxopentan-2-yl]morpholine-4-carboxamide |
NA |
107000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSS |
Morpholine-4-carboxylic acid [1-(1-cyano-3-phenyl-propylcarbamoyl)-ethyl]-amide |
NA |
134000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSS |
Benzyl 1-((cyanomethyl)carbamoyl)cyclopentylcarbamate |
150000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CTSS |
N-[1-(cyanomethylcarbamoyl)cyclohexyl]-4-(4-methylpiperazine-1-carbonyl)benzamide |
110000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CTSS |
N-[1-(cyanomethylcarbamoyl)cyclohexyl]-4-(4-methylpiperazin-1-yl)sulfonylbenzamide |
102000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CTSS |
Ac-Glu(OtBu)-Ala-LeuVSMe |
NA |
170000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSS |
pTosyl-NeopentylAsn-Ser-LeuVSMe |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| CTSS |
Benzyl 1-((cyanomethyl)carbamoyl)cyclopropylcarbamate |
150000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CTSS |
benzyl N-[(2S)-1-(cyanomethylamino)-3,3-dimethyl-1-oxobutan-2-yl]carbamate |
150000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CTSS |
Morpholine-4-carboxylic acid [3-methyl-1-(1-methyl-3-phenyl-propylcarbamoyl)-butyl]-amide |
NA |
339000 |
NA |
NA |
NA |
NA |
TTD |
| CTSS |
tert-butyl N-{[(cyanomethyl)carbamoyl]methyl}carbamate |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CTSS |
Carbamic acid, [2-[(cyanomethyl)amino]-1-methyl-2-oxoethyl]-, 1,1-dimethylethyl ester, (s)- |
292000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSS |
benzyl N-{[(cyanomethyl)carbamoyl]methyl}carbamate |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CTSS |
Cathepsin X-IN-1 |
NA |
241000 |
NA |
NA |
NA |
NA |
BindingDB |
| CTSS |
7-[3-(4-chlorophenoxy)-2-hydroxypropyl]-3-methyl-8-sulfanyl-3,7-dihydro-1H-purine-2,6-dione |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CTSS |
1-benzyl-3,7-dimethyl-8-sulfanylidene-9H-purine-2,6-dione |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CTSS |
2-((2S,3S)-2-Acetoxy-4-oxo-azetidin-3-ylcarbamoyl)-pyrrolidine-1-carboxylic acid benzyl ester |
150000 |
NA |
NA |
NA |
NA |
NA |
TTD |