| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CTSS |
tert-butyl N-[(2S)-1-oxo-1-(5-propan-2-yl-1,3,4-oxadiazol-2-yl)pentan-2-yl]carbamate |
130000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CTSS |
1-ethyl-8-mercapto-3,7-dimethyl-1H-purine-2,6(3H,7H)-dione |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CTSS |
Caffeine, 8-mercapto- |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| CTSV |
(1r)-1-{[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]methyl}-2,2-dimethylpropyl(1S)-1-[oxo(1h-pyrazol-5-ylamino)acetyl]pentylcarbamate |
NA |
230000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CXCL12 |
2-[[4-(Carboxymethylsulfanyl)-6-phenyl-1,3,5-triazin-2-yl]oxy]acetic acid |
NA |
NA |
200000 |
NA |
NA |
NA |
BindingDB |
| CXCL12 |
CXCL12 ligand 1 |
NA |
NA |
234000 |
NA |
NA |
NA |
BindingDB |
| CXCL12 |
2-[[4-(Carboxymethylsulfanyl)-6-pyrrolidin-1-yl-1,3,5-triazin-2-yl]sulfanyl]acetic acid |
NA |
NA |
1030000 |
NA |
NA |
NA |
BindingDB |
| CXCL12 |
2-[[4-(Carboxymethylsulfanyl)-6-(3-oxa-8-azabicyclo[3.2.1]octan-8-yl)-1,3,5-triazin-2-yl]sulfanyl]acetic acid |
NA |
NA |
233000 |
NA |
NA |
NA |
BindingDB |
| CXCL12 |
2-[[4-(Carboxymethylamino)-6-phenyl-1,3,5-triazin-2-yl]amino]acetic acid |
NA |
NA |
355000 |
NA |
NA |
NA |
BindingDB |
| CXCL12 |
2-[[4-(Carboxymethylsulfanyl)-6-thiophen-3-yl-1,3,5-triazin-2-yl]sulfanyl]acetic acid |
NA |
NA |
1344000 |
NA |
NA |
NA |
BindingDB |
| CXCL12 |
2-[[4-[3,5-Bis(trifluoromethyl)phenyl]-6-(carboxymethylsulfanyl)-1,3,5-triazin-2-yl]sulfanyl]acetic acid |
NA |
NA |
646000 |
NA |
NA |
NA |
BindingDB |
| CXCL12 |
2-[[4-(Carboxymethylsulfanyl)-6-thiophen-2-yl-1,3,5-triazin-2-yl]sulfanyl]acetic acid |
NA |
NA |
1640000 |
NA |
NA |
NA |
BindingDB |
| CXCL12 |
2-[[4-Anilino-6-(carboxymethylsulfanyl)-1,3,5-triazin-2-yl]sulfanyl]acetic acid |
NA |
NA |
251000 |
NA |
NA |
NA |
BindingDB |
| CXCL12 |
2-[[4-(Carboxymethylsulfanyl)-6-(4-methylmorpholin-4-ium-4-yl)-1,3,5-triazin-2-yl]sulfanyl]acetic acid;chloride |
NA |
NA |
3024000 |
NA |
NA |
NA |
BindingDB |
| CXCL12 |
(2S)-2-[[4-[[(1R)-1-carboxypentyl]amino]-6-phenyl-1,3,5-triazin-2-yl]amino]hexanoic acid |
NA |
NA |
383000 |
NA |
NA |
NA |
BindingDB |
| CXCL12 |
2-[[4-(Carboxymethylsulfanyl)-6-(3-hydroxyphenyl)-1,3,5-triazin-2-yl]sulfanyl]acetic acid |
NA |
NA |
1798000 |
NA |
NA |
NA |
BindingDB |
| CXCL12 |
(2S)-2-[[4-[[(1S)-1-carboxypentyl]amino]-6-phenyl-1,3,5-triazin-2-yl]amino]hexanoic acid |
NA |
NA |
156000 |
NA |
NA |
NA |
BindingDB |
| CXCL12 |
2-[[4-(Carboxymethylsulfanyl)-6-(cyclohexylamino)-1,3,5-triazin-2-yl]sulfanyl]acetic acid |
NA |
NA |
170000 |
NA |
NA |
NA |
BindingDB |
| CXCL12 |
3-[4,6-Bis(carboxymethylsulfanyl)-1,3,5-triazin-2-yl]benzoic acid |
NA |
NA |
133000 |
NA |
NA |
NA |
BindingDB |
| CXCL12 |
2-[[4-(Carboxymethylsulfanyl)-6-phenyl-1,3,5-triazin-2-yl]sulfanyl]acetic acid |
NA |
NA |
158000 |
NA |
NA |
NA |
BindingDB |