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negative DTIs
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Drugs And Genes
Negative Drug Target Genes
Gene
Drug
GENE_SYMBOL
DRUG_NAME
Ki (nM)
IC50 (nM)
Kd (nM)
EC50 (nM)
Potency (nM)
AC50 (nM)
Datasource
CXCR1
Ac-Leu-Asn-Phe-Thr-Gly-Met-Pro-Pro-Ala-Asp-Glu-Asp-Tyr-Ser-Pro-NH2
3100000
NA
NA
NA
NA
NA
TTD
CXCR1
Ac-Phe-Thr-Gly-Met-Pro-Pro-Ala-Asp-Glu-Asp-Tyr-Ser-Pro-NH2
1850000
NA
NA
NA
NA
NA
TTD
CXCR1
Ac-Gly-Met-Pro-Pro-Ala-Asp-Glu-Asp-Tyr-Ser-Pro-NH2
890000
NA
NA
NA
NA
NA
TTD
CXCR1
Ac-Met-Trp-Asp-Phe-Asp-Asp-Leu-Asn-Phe-Thr-Gly-Met-Ala-Pro-Ala-Asp-Glu-Asp-Tyr-Ser-Pro-NH2
400000
NA
NA
NA
NA
NA
TTD
CXCR1
Ac-Met-Trp-Asp-Phe-Asp-Asp-Leu-Asn-Phe-Thr-Gly-Met-Pro-Pro-Ala-Asp-Glu-Asp-Ala-Ser-Pro-NH2
265000
NA
NA
NA
NA
NA
TTD
CXCR1
Ac-Met-Trp-Asp-Phe-Asp-Asp-Leu-Asn-Phe-Thr-Gly-Met-Pro-Pro-Ala-Asp-Glu-Asp-Tyr-Ser-Ala-NH2
155000
NA
NA
NA
NA
NA
TTD
CXCR1
Ac-Met-Trp-Asp-Phe-Asp-Asp-Leu-Asn-Ala-Thr-Gly-Met-Pro-Pro-Ala-Asp-Glu-Asp-Tyr-Ser-Pro-NH2
107000
NA
NA
NA
NA
NA
TTD
CXCR1
Ac-Thr-Gly-Met-Pro-Pro-Ala-Asp-Glu-Asp-Tyr-Ser-Pro-NH2
2050000
NA
NA
NA
NA
NA
TTD
CXCR1
Ac-Asn-Phe-Thr-Gly-Met-Pro-Pro-Ala-Asp-Glu-Asp-Tyr-Ser-Pro-NH2
2700000
NA
NA
NA
NA
NA
TTD
CXCR2
Ac-Phe-Asp-Asp-Leu-Asn-Phe-Thr-Gly-Met-Pro-Pro-Ala-Asp-Glu-Asp-Tyr-Ser-Pro-NH2
120000
NA
NA
NA
NA
NA
BindingDB|TTD
CXCR2
Ac-Asp-Asp-Leu-Asn-Phe-Thr-Gly-Met-Pro-Pro-Ala-Asp-Glu-Asp-Tyr-Ser-Pro-NH2
190000
NA
NA
NA
NA
NA
BindingDB|TTD
CXCR2
Ac-Asp-Leu-Asn-Phe-Thr-Gly-Met-Pro-Pro-Ala-Asp-Glu-Asp-Tyr-Ser-Pro-NH2
750000
NA
NA
NA
NA
NA
BindingDB|TTD
CXCR2
Ac-Leu-Asn-Phe-Thr-Gly-Met-Pro-Pro-Ala-Asp-Glu-Asp-Tyr-Ser-Pro-NH2
3100000
NA
NA
NA
NA
NA
BindingDB|TTD
CXCR2
Ac-Phe-Thr-Gly-Met-Pro-Pro-Ala-Asp-Glu-Asp-Tyr-Ser-Pro-NH2
1850000
NA
NA
NA
NA
NA
BindingDB|TTD
CXCR2
Ac-Gly-Met-Pro-Pro-Ala-Asp-Glu-Asp-Tyr-Ser-Pro-NH2
890000
NA
NA
NA
NA
NA
BindingDB|TTD
CXCR2
Ac-Met-Trp-Asp-Phe-Asp-Asp-Leu-Asn-Phe-Thr-Gly-Met-Ala-Pro-Ala-Asp-Glu-Asp-Tyr-Ser-Pro-NH2
400000
NA
NA
NA
NA
NA
BindingDB|TTD
CXCR2
Ac-Met-Trp-Asp-Phe-Asp-Asp-Leu-Asn-Phe-Thr-Gly-Met-Pro-Pro-Ala-Asp-Glu-Asp-Ala-Ser-Pro-NH2
265000
NA
NA
NA
NA
NA
BindingDB|TTD
CXCR2
Ac-Met-Trp-Asp-Phe-Asp-Asp-Leu-Asn-Phe-Thr-Gly-Met-Pro-Pro-Ala-Asp-Glu-Asp-Tyr-Ser-Ala-NH2
155000
NA
NA
NA
NA
NA
BindingDB|TTD
CXCR2
Ac-Met-Trp-Asp-Phe-Asp-Asp-Leu-Asn-Ala-Thr-Gly-Met-Pro-Pro-Ala-Asp-Glu-Asp-Tyr-Ser-Pro-NH2
107000
NA
NA
NA
NA
NA
BindingDB|TTD
CXCR2
Ac-Thr-Gly-Met-Pro-Pro-Ala-Asp-Glu-Asp-Tyr-Ser-Pro-NH2
2050000
NA
NA
NA
NA
NA
BindingDB|TTD
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