| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CXCR2 |
Ac-Asn-Phe-Thr-Gly-Met-Pro-Pro-Ala-Asp-Glu-Asp-Tyr-Ser-Pro-NH2 |
2700000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CXCR4 |
US9205085, Msx-164 |
NA |
NA |
NA |
5011872.34 |
NA |
NA |
TTD |
| CXCR4 |
1,4-Bis-(1-anilinoethyl) benzene |
NA |
NA |
NA |
19952623.15 |
NA |
NA |
TTD |
| CXCR4 |
US9205085, Msx-172 |
NA |
NA |
NA |
100000000 |
NA |
NA |
TTD |
| CXCR4 |
US9205085, Msx-183 |
NA |
NA |
NA |
1000000000 |
NA |
NA |
TTD |
| CXCR4 |
4-nitro-N-(4-{[(4-nitrophenyl)amino]methyl}benzyl)aniline |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| CXCR4 |
US9205085, Msx-184 |
NA |
NA |
NA |
10000000 |
NA |
NA |
TTD |
| CXCR4 |
US9205085, Msx-205 |
NA |
NA |
NA |
1000000000 |
NA |
NA |
TTD |
| CXCR4 |
N,N'-Bis(3-methoxyphenyl)terephthalamide |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| CXCR4 |
4-methyl-N-[4-(4-toluidinomethyl)benzyl]aniline |
NA |
NA |
NA |
100000000 |
NA |
NA |
TTD |
| CXCR4 |
N-(4-{[3-(trifluoromethyl)anilino]methyl}benzyl)-N-[3-(trifluoromethyl)phenyl]amine |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| CXCR4 |
N,N'-(1,4-Phenylenedimethylidyne)DI-P-anisidine |
NA |
NA |
NA |
39810717.06 |
NA |
NA |
TTD |
| CXCR4 |
US9205085, Msx-173 |
NA |
NA |
NA |
5011872.34 |
NA |
NA |
TTD |
| CXCR4 |
alpha,alpha'-Bis(4-fluoroanilino)-P-xylene |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| CXCR4 |
US9205085, Msx-206 |
NA |
NA |
NA |
100000000 |
NA |
NA |
TTD |
| CXCR4 |
US9205085, Msx-203 |
NA |
NA |
NA |
1000000000 |
NA |
NA |
TTD |
| CYB5R3 |
Propylthiouracil |
NA |
279400 |
NA |
NA |
NA |
NA |
PubChem |
| CYP11B1 |
3-(6-Chloro-pyridin-3-yl)-6,6-dimethyl-3,5,6,7-tetrahydro-benzoimidazol-4-one |
NA |
6900000 |
NA |
NA |
NA |
NA |
BindingDB |
| CYP11B1 |
3-(3,4-Dichloro-phenyl)-6,6,-dimethyl-3,5,6,7-tetrahydro-benzoimidazol-4-one |
NA |
370000 |
NA |
NA |
NA |
NA |
BindingDB |
| CYP11B1 |
3-(1-Methyl-2-oxo-3,4-dihydroquinolin-6-yl)spiro[5,7-dihydrobenzimidazole-6,1''-cyclobutane]-4-one |
NA |
14000000 |
NA |
NA |
NA |
NA |
BindingDB |