| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CXCL12 |
2-[[4-(Carboxymethylsulfanyl)-6-(4-morpholin-4-ylphenyl)-1,3,5-triazin-2-yl]sulfanyl]acetic acid |
NA |
NA |
306000 |
NA |
NA |
NA |
BindingDB |
| CXCL12 |
3-[[4-(2-Carboxyethylsulfanyl)-6-phenyl-1,3,5-triazin-2-yl]sulfanyl]propanoic acid |
NA |
NA |
158000 |
NA |
NA |
NA |
BindingDB |
| CXCL12 |
2-[[4-(Carboxymethylsulfanyl)-6-(4-methoxyphenyl)-1,3,5-triazin-2-yl]sulfanyl]acetic acid |
NA |
NA |
357000 |
NA |
NA |
NA |
BindingDB |
| CXCL12 |
2-[[4-(1-Bicyclo[1.1.1]pentanylamino)-6-(carboxymethylsulfanyl)-1,3,5-triazin-2-yl]sulfanyl]acetic acid |
NA |
NA |
1355000 |
NA |
NA |
NA |
BindingDB |
| CXCL12 |
[(6-Phenylpyrimidin-4-yl)thio]acetic acid |
NA |
NA |
900000 |
NA |
NA |
NA |
BindingDB |
| CXCL12 |
2-({2-[(Carboxymethyl)sulfanyl]-6-phenylpyrimidin-4-yl}sulfanyl)acetic acid |
NA |
NA |
169000 |
NA |
NA |
NA |
BindingDB |
| CXCL12 |
2-[2-(Carboxymethylsulfanyl)-6-methylpyrimidin-4-yl]sulfanylacetic acid |
NA |
NA |
1200000 |
NA |
NA |
NA |
BindingDB |
| CXCL12 |
{4-[(3,4-Dimethylphenyl)sulfamoyl]-2-methylphenoxy}acetic acid |
NA |
NA |
4100000 |
NA |
NA |
NA |
BindingDB |
| CXCL12 |
[(4-Fluoroanilino)-(4-propoxyphenyl)methyl]phosphonic acid;propan-2-ol |
NA |
NA |
1100000 |
NA |
NA |
NA |
BindingDB |
| CXCL12 |
2-[2-[(3-fluorophenyl)carbamoyl]-3,4-dihydro-1H-isoquinolin-1-yl]acetic acid |
NA |
NA |
4100000 |
NA |
NA |
NA |
BindingDB |
| CXCL12 |
(2S)-2-[3-(4-chloroindol-1-yl)propanoylamino]propanoic acid |
NA |
NA |
1700000 |
NA |
NA |
NA |
BindingDB |
| CXCL12 |
(E)-1-(4'-Chlorophenyl)-3-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-one |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB |
| CXCL12 |
N-[(9,10-dioxo-9,10-dihydroanthracen-2-yl)sulfonyl]glycine |
NA |
NA |
1200000 |
NA |
NA |
NA |
BindingDB |
| CXCL12 |
nonasodium;(2R,3S,4S,5R,6R)-6-[(2R,3S,4R,5R,6R)-6-[(2R,3S,4S,5R,6R)-6-[(2R,3S,4R,5R,6R)-6-[(2R,3S,4S,5R,6R)-6-[(2R,3S,4R,5R,6S)-6-(5-aminopentoxy)-4-hydroxy-2-(hydroxymethyl)-5-(sulfonatoamino)oxan-3-yl]oxy-2-carboxylato-4-hydroxy-5-sulfonatooxyoxan-3-yl]oxy-4-hydroxy-2-(hydroxymethyl)-5-(sulfonatoamino)oxan-3-yl]oxy-2-carboxylato-4-hydroxy-5-sulfonatooxyoxan-3-yl]oxy-4-hydroxy-2-(hydroxymethyl)-5-(sulfonatoamino)oxan-3-yl]oxy-3,4-dihydroxy-5-sulfonatooxyoxane-2-carboxylate |
NA |
NA |
250000000 |
NA |
NA |
NA |
BindingDB |
| CXCL8 |
Interleukin-8 inhibitor, 6 |
106000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CXCL8 |
Interleukin-8 inhibitor, 4 |
383000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CXCL8 |
Phenazopyridine Hydrochloride |
NA |
NA |
NA |
NA |
118832 |
NA |
PubChem |
| CXCR1 |
Ac-Phe-Asp-Asp-Leu-Asn-Phe-Thr-Gly-Met-Pro-Pro-Ala-Asp-Glu-Asp-Tyr-Ser-Pro-NH2 |
120000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CXCR1 |
Ac-Asp-Asp-Leu-Asn-Phe-Thr-Gly-Met-Pro-Pro-Ala-Asp-Glu-Asp-Tyr-Ser-Pro-NH2 |
190000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CXCR1 |
Ac-Asp-Leu-Asn-Phe-Thr-Gly-Met-Pro-Pro-Ala-Asp-Glu-Asp-Tyr-Ser-Pro-NH2 |
750000 |
NA |
NA |
NA |
NA |
NA |
TTD |