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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
DPP4 N-(1,3-benzodioxol-5-ylmethyl)-N-(2-piperidin-1-yl-2-thioxoethyl)amine NA 1000000 NA NA NA NA TTD
DPP4 diphenyl 1-((2S,3S)-2-amino-3-methylpentanoyl)pyrrolidin-2-ylphosphonate NA 125000 NA NA NA NA TTD
DPP4 N-((S)-3-Amino-4-oxo-4-piperidin-1-yl-butyl)-acetamide NA 518000 NA NA NA NA BindingDB|TTD
DPP4 2-Cyclohexylamino-1-piperidin-1-yl-propan-1-one NA 217000 NA NA NA NA BindingDB|TTD
DPP4 (S)-2,5-Diamino-1-piperidin-1-yl-pentane-1-thione NA 1000000 NA NA NA NA TTD
DPP4 (S)-2-Amino-4-(4-chloro-benzylamino)-1-(4-methyl-piperidin-1-yl)-butan-1-one NA 500000 NA NA NA NA TTD
DPP4 (S)-2,6-diamino-1-(piperidin-1-yl)hexan-1-one NA 247000 NA NA NA NA BindingDB|TTD
DPP4 (2S)-2-amino-1-(2-diphenoxyphosphorylpyrrolidin-1-yl)-3-phenyl-propan-1-one NA 142000 NA NA NA NA BindingDB|TTD
DPP4 (2S)-2-amino-3-(1H-indol-3-yl)-1-pyrrolidin-1-ylpropan-1-one NA 286000 NA NA NA NA BindingDB|TTD
DPP4 (2S,3S)-2-amino-1-(azepan-1-yl)-3-methylpentan-1-one NA 374000 NA NA NA NA BindingDB|TTD
DPP4 (2S,3S)-2-amino-1-(3-azidopyrrolidin-1-yl)-3-methylpentan-1-one NA 107000 NA NA NA NA BindingDB|TTD
DPP4 (2S,3S)-2-amino-N-cyclopentyl-3-methylpentanamide NA 1000000 NA NA NA NA TTD
DPP4 2-(Adamantan-1-ylamino)-1-(3-hydroxy-pyrrolidin-1-yl)-ethanone NA 1000000 NA NA NA NA TTD
DPP4 (2Z)-2-{1-fluoro-2-[(2-phenylethyl)amino]ethylidene}cyclopentane-1-carbonitrile NA 500000 NA NA NA NA TTD
DPP4 1-[2-(Cyclohexyl-methyl-amino)-acetyl]-pyrrolidine-2-carbonitrile NA 103000 NA NA NA NA BindingDB|TTD
DPP4 (2S)-1-[2-[2-[(5-cyanopyridin-2-yl)amino]ethylamino]acetyl]pyrrolidine-2-carboxamide NA 434000 NA NA NA NA BindingDB|TTD
DPP4 (2S)-2,4-diamino-N-[cyclohexyl(diphenoxyphosphoryl)methyl]butanamide NA 1000000 NA NA NA NA BindingDB
DPP4 1-[2-(3-Hydroxy-adamantan-1-ylamino)-acetyl]-pyrrolidine-2-carboxylic acid NA 477000 NA NA NA NA BindingDB|TTD
DPP4 (2E)-2-(1-fluoro-2-{[(4-fluorophenyl)methyl]amino}ethylidene)cyclopentane-1-carbonitrile NA 500000 NA NA NA NA TTD
DPP4 (3S)-3-amino-4-(2-diphenoxyphosphorylpyrrolidin-1-yl)-4-oxo-butanoic Acid NA 1000000 NA NA NA NA TTD