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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
DPP4 (2S)-2-amino-1-(2-diphenoxyphosphorylpyrrolidin-1-yl)-3-(1H-imidazol-4-yl)propan-1-one NA 326000 NA NA NA NA BindingDB|TTD
DPP4 1-[2-(1H-Benzoimidazol-2-ylamino)-acetyl]-pyrrolidine-2-carbonitrile NA 1000000 NA NA NA NA TTD
DPP4 1-[2-(3-Hydroxy-adamantan-1-ylamino)-acetyl]-pyrrolidine-2-carboxylic acid amide NA 931000 NA NA NA NA BindingDB|TTD
DPP4 (2Z)-2-(1-fluoro-2-{[(4-fluorophenyl)methyl]amino}ethylidene)cyclopentane-1-carbonitrile NA 1000000 NA NA NA NA TTD
DPP4 1-(3-Cyclohexyl-propionyl)-pyrrolidine-2-carbonitrile NA 500000 NA NA NA NA TTD
DPP4 (2E)-2-{1-fluoro-2-[(2-phenylethyl)amino]ethylidene}cyclopentane-1-carbonitrile NA 1000000 NA NA NA NA TTD
DPP4 2-(S)-Amino-4-(2-methoxy-benzylamino)-1-piperidin-1-yl-butan-1-one NA 500000 NA NA NA NA TTD
DPP4 (S)-2-Amino-4-[bis-(4-chloro-benzyl)-amino]-1-piperidin-1-yl-butan-1-one NA 125000 NA NA NA NA TTD
DPP4 2-Oxo-2-pyrrolidin-1-ylethanamine NA 1000000 NA NA NA NA TTD
DPP4 (S)-3-amino-4-oxo-4-(pyrrolidin-1-yl)butanoic acid NA 122000 NA NA NA NA BindingDB
DPP4 (2H-1,3-benzodioxol-5-ylmethyl)(2-cyclopentylideneethyl)amine NA 250000 NA NA NA NA TTD
DPP4 (2S)-2-amino-4-(naphthalen-1-ylmethylamino)-1-piperidin-1-ylbutan-1-one NA 301000 NA NA NA NA BindingDB|TTD
DPP4 2-(S)-Amino-4-(3-methoxy-benzylamino)-1-piperidin-1-yl-butan-1-one NA 250000 NA NA NA NA BindingDB|TTD
DPP4 (S)-3-amino-4-oxo-4-(pyrrolidin-1-yl)butanamide NA 188000 NA NA NA NA BindingDB|TTD
DPP4 (S)-1-((S)-2,4-Diamino-butyryl)-piperidine-2-carbonitrile NA 151000 NA NA NA NA BindingDB|TTD
DPP4 N-Cyclohexyl-2-oxo-2-(1-pyrrolidinyl)ethaneamine NA 148000 NA NA NA NA BindingDB|TTD
DPP4 2-(S)-Amino-4-(2-chloro-benzylamino)-1-piperidin-1-yl-butan-1-one NA 345000 NA NA NA NA BindingDB|TTD
DPP4 N4-(4-chlorobenzyl)-2,4-diaminobutanoylpiperidine NA 165000|196000 NA NA NA NA BindingDB
DPP4 (2S)-2-amino-4-(naphthalen-2-ylmethylamino)-1-piperidin-1-ylbutan-1-one NA 179000 NA NA NA NA BindingDB|TTD
DPP4 (2S)-2-amino-4-[(4-chlorophenyl)methylamino]-1-(4-hydroxypiperidin-1-yl)butan-1-one NA 1000000 NA NA NA NA TTD