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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
DPP4 2-(S)-Amino-4-(4-methoxy-benzylamino)-1-piperidin-1-yl-butan-1-one NA 417000 NA NA NA NA BindingDB|TTD
DPP4 2-(S)-Amino-4-(cyclohexylmethyl-amino)-1-piperidin-1-yl-butan-1-one NA 496000 NA NA NA NA BindingDB|TTD
DPP4 N-(1,3-benzodioxol-5-ylmethyl)-N-(2-oxo-2-pyrrolidin-1-ylethyl)amine NA 1000000 NA NA NA NA TTD
DPP4 6-((S)-3-Amino-4-oxo-4-piperidin-1-yl-butylamino)-nicotinonitrile NA 205000 NA NA NA NA BindingDB|TTD
DPP4 (S)-2-Amino-4-(4-chloro-benzylamino)-1-(3,6-dihydro-2H-pyridin-1-yl)-butan-1-one NA 148000 NA NA NA NA BindingDB|TTD
DPP4 N-((S)-3-Amino-4-oxo-4-piperidin-1-yl-butyl)-benzamide NA 418000 NA NA NA NA BindingDB|TTD
DPP4 (S)-2-amino-3-hydroxy-1-(pyrrolidin-1-yl)propan-1-one NA 190000 NA NA NA NA BindingDB|TTD
DPP4 (2S)-2,6-diamino-1-(3-hydroxypyrrolidin-1-yl)hexan-1-one NA 500000 NA NA NA NA BindingDB|TTD
DPP4 (2S)-2-amino-1-piperidin-1-yl-4-(thiophen-2-ylmethylamino)butan-1-one NA 278000 NA NA NA NA BindingDB|TTD
DPP4 2-(S)-Amino-4-(3-phenyl-propylamino)-1-piperidin-1-yl-butan-1-one NA 500000 NA NA NA NA TTD
DPP4 (2S)-2-amino-1-piperidin-1-yl-4-(pyridin-4-ylmethylamino)butan-1-one NA 125000 NA NA NA NA BindingDB|TTD
DPP4 N-Benzyl-2-oxo-2-(1-pyrrolidinyl)ethaneamine NA 1000000 NA NA NA NA BindingDB|TTD
DPP4 (S)-2-Amino-4-(4-chloro-benzylamino)-1-(2-methyl-piperidin-1-yl)-butan-1-one NA 500000 NA NA NA NA TTD
DPP4 (2S)-2-amino-4-[(4-phenylmethoxyphenyl)methylamino]-1-piperidin-1-ylbutan-1-one NA 192000 NA NA NA NA BindingDB|TTD
DPP4 (S)-2-Amino-4-(4-chloro-benzylamino)-1-(3-methyl-piperidin-1-yl)-butan-1-one NA 500000 NA NA NA NA TTD
DPP4 2-(S)-Amino-4-(2-benzyloxy-benzylamino)-1-piperidin-1-yl-butan-1-one NA 500000 NA NA NA NA TTD
DPP4 2-(S)-Amino-4-(3-chloro-benzylamino)-1-piperidin-1-yl-butan-1-one NA 186000 NA NA NA NA BindingDB|TTD
DPP4 (S)-2-Amino-4-phenylamino-1-piperidin-1-yl-butan-1-one NA 250000 NA NA NA NA BindingDB|TTD
DPP4 2-(S)-Amino-4-cyclohexylamino-1-piperidin-1-yl-butan-1-one NA 1000000 NA NA NA NA TTD
DPP4 2-(S)-Amino-4-phenethylamino-1-piperidin-1-yl-butan-1-one NA 188000 NA NA NA NA BindingDB|TTD