| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| DPP4 |
US11096924, DASH-inhibitors 5323 |
NA |
60270000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP4 |
(S)-2,5-diamino-1-(pyrrolidin-1-yl)pentan-1-one |
NA |
118000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP4 |
(S)-benzyl 5-amino-6-(3,4-dihydroquinolin-1(2H)-yl)-6-oxohexylcarbamate |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| DPP4 |
US11096924, DASH-inhibitors 5322 |
NA |
9818000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP4 |
US11096924, DASH-inhibitors 5333 |
NA |
4426000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP4 |
US11096924, DASH-inhibitors 5321 |
NA |
20270000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP4 |
US11096924, DASH-inhibitors 1049 C |
NA |
830000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP4 |
US11096924, DASH-inhibitors 4160 |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP4 |
7-(2-Hydroxyethylamino)-6-nitro-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one |
NA |
121300 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP4 |
H-Gly-Ile-Pro-Leu-Pro-Leu-Ile-OH |
NA |
3830000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP4 |
(R)-1-(2-pivalamidoacetyl)pyrrolidin-2-ylboronic acid |
608000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP4 |
(2S,4S)-4-(4-chlorobenzylamino)-2-amino-1-(piperidin-1-yl)pentan-1-one |
NA |
325000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP4 |
H-Tyr-Pro-Ala-NH2 |
170000|420000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP4 |
Tyr-Pro-Ala |
270000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| DPP4 |
N-[4-[2-(2,3-dihydro-1,4-benzodioxin-3-ylmethylamino)ethoxy]phenyl]-2-methylpropane-1-sulfonamide;hydrochloride |
NA |
326600 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP4 |
4-[3-Azido-3-(2,3-dihydro-1,4-benzodioxin-3-yl)propoxy]benzenesulfonamide |
NA |
669300 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP4 |
N-[4-[2-(2,3-dihydro-1,4-benzodioxin-3-ylmethylamino)ethoxy]phenyl]methanesulfonamide;hydrochloride |
NA |
300200 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP4 |
4-[3-Azido-3-(2,3-dihydro-1,4-benzodioxin-3-yl)propoxy]-3-methoxybenzenesulfonamide |
NA |
326600 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP4 |
CID 171345933 |
NA |
620000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP4 |
(2S)-2-Amino-2-cyclohexyl-1-(1,3-dihydro-2H-isoindol-2-YL)ethanone |
NA |
1375000 |
NA |
NA |
NA |
NA |
BindingDB |