| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| DPP4 |
N-(1,3-benzodioxol-5-ylmethyl)-2-cyclohexylidene-2-fluoroethanamine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| DPP4 |
(2-Cyclohexylidene-2-fluoroethyl)[(4-fluorophenyl)methyl]amine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| DPP4 |
(2-Cyclohexylidene-2-fluoroethyl)({[3-(trifluoromethyl)phenyl]methyl})amine |
NA |
125000 |
NA |
NA |
NA |
NA |
TTD |
| DPP4 |
(2-Cyclohexylidene-2-fluoroethyl)(2-phenylethyl)amine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| DPP4 |
N-(2-cyclohexylidene-2-fluoroethyl)piperidin-4-amine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| DPP4 |
1-Benzyl-N-(2-cyclohexylidene-2-fluoroethyl)-4-piperidinamine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| DPP4 |
(2-Cyclohexylidene-2-fluoroethyl)[3-(dimethylamino)propyl]amine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| DPP4 |
N-(2-cyclopentylideneethyl)cyclohexanamine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| DPP4 |
Benzyl(2-cyclopentylideneethyl)amine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| DPP4 |
diphenyl 2-((S)-2,6-diaminohexanoyl)isoindolin-1-ylphosphonate |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| DPP4 |
diphenyl 2-((2S,3R)-2-amino-3-methylpentanoyl)isoindolin-1-ylphosphonate |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| DPP4 |
di-(4-acetamido)phenyl 2-((S)-2,6-diaminohexanoyl)isoindolin-1-ylphosphonate |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| DPP4 |
di-(4-acetamido)phenyl 2-((2S,3S)-2-amino-3-methylpentanoyl)isoindolin-1-ylphosphonate |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| DPP4 |
diphenyl 2-((2S,3S)-2-amino-3-methylpentanoyl)isoindolin-1-ylphosphonate |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| DPP4 |
di-(4-acetamido)phenyl 2-((2S,3R)-2-amino-3-methylpentanoyl)isoindolin-1-ylphosphonate |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| DPP4 |
N-Cyclopentyl L-isoleucinamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| DPP4 |
2-Amino-1-azepan-1-yl-3-methyl-pentan-1-one |
NA |
374000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP4 |
2-amino-N,N,3-trimethylpentanamide |
NA |
360000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP4 |
(2S,3R)-2-amino-1-(5-fluoroisoindolin-2-yl)-3-methylpentan-1-one |
NA |
7900000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP4 |
2,4-Diamino-1-piperidin-1-yl-butan-1-one |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |