| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| DPP4 |
N-benzyl-2-(1-pyrrolidinyl)ethanamine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| DPP4 |
N-(1,3-benzodioxol-5-ylmethyl)-2-pyrrolidin-1-ylethanamine |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| DPP4 |
N-(2-pyrrolidin-1-ylethyl)cyclohexanamine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| DPP4 |
2-Amino-3-methyl-pentanoic acid methyl-propyl-amide |
NA |
377000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP4 |
2-Amino-1-piperidin-1-yl-pentan-1-one |
NA |
229000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP4 |
1-Aminomethyl-6,7-dimethoxy-isoquinoline-4-carboxylic acid; hydrochloride |
NA |
103000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP4 |
1-Dimethylaminomethyl-6,7-dimethoxy-isoquinoline-4-carboxylic acid ethyl ester; hydrochloride |
NA |
948000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP4 |
1-Aminomethyl-6,7-dimethoxy-isoquinoline-4-carbaldehyde; hydrochloride |
NA |
277000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP4 |
1-(2-Amino-ethyl)-6,7-dimethoxy-isoquinoline-4-carboxylic acid ethyl ester; TFA |
NA |
746000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP4 |
1-Aminomethyl-6,7-dimethoxy-isoquinoline-4-carboxylic acid amide; hydrochloride |
NA |
170000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP4 |
2-Amino-3-[2-(2-cyano-pyrrolidin-1-yl)-2-oxo-ethylamino]-2-methyl-propionic acid |
NA |
109000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP4 |
2-Amino-3-(1H-imidazol-4-yl)-1-piperidin-1-yl-propan-1-one |
NA |
213000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP4 |
Pyrrolidin-2-yl-pyrrolidin-1-yl-methanethione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| DPP4 |
2-Amino-1-piperidin-1-yl-hexan-1-one |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP4 |
2-Amino-2-cyclohexyl-1-piperidin-1-yl-ethanone |
NA |
217000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP4 |
Benzoic acid 1-(2,6-diamino-hexanoyl)-pyrrolidin-3-yl ester |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| DPP4 |
2,6-Diamino-1-azetidin-1-yl-hexan-1-one |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP4 |
2,6-Diamino-1-azepan-1-yl-hexan-1-one |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| DPP4 |
Pyrrolidin-1-yl-(tetrahydro-thiophen-2-yl)-methanone |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| DPP4 |
2,6-Diamino-1-(3,6-dihydro-2H-pyridin-1-yl)-hexan-1-one |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |