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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
DPP4 2-Amino-3-methyl-pentanoic acid diethylamide NA 500000 NA NA NA NA TTD
DPP4 [5-Amino-1-(piperidine-1-carbonyl)-pentyl]-carbamic acid benzyl ester NA 134900 NA NA NA NA BindingDB|TTD
DPP4 2,6-Diamino-1-piperidin-1-yl-hexan-1-one NA 247000 NA NA NA NA BindingDB|TTD
DPP4 2-Amino-3-hydroxy-1-pyrrolidin-1-yl-propan-1-one NA 190000 NA NA NA NA BindingDB|TTD
DPP4 2-Amino-3-methyl-pentanoic acid ethyl-methyl-amide NA 167000 NA NA NA NA BindingDB|TTD
DPP4 5-(Aminomethyl)-2-phenyl-6-[3-(trifluoromethyl)phenyl]pyrimidin-4-amine NA 170000 NA NA NA NA BindingDB|TTD
DPP4 (2S)-2-amino-2-cyclohexyl-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one NA 230000 NA NA NA NA BindingDB
DPP4 N-(2-cyclopentylidene-2-fluoroethyl)cyclohexanamine NA 1000000 NA NA NA NA TTD
DPP4 Benzyl(2-cyclopentylidene-2-fluoroethyl)amine NA 1000000 NA NA NA NA TTD
DPP4 (2-Cyclopentylidene-2-fluoroethyl)[(4-methoxyphenyl)methyl]amine NA 1000000 NA NA NA NA TTD
DPP4 (2-Cyclopentylidene-2-fluoroethyl)[(4-fluorophenyl)methyl]amine NA 1000000 NA NA NA NA TTD
DPP4 N-(2-Cyclopentylidene-2-fluoroethyl)-N-(2-pyridinylethyl)amine NA 1000000 NA NA NA NA TTD
DPP4 (2-Cyclopentylidene-2-fluoroethyl)(2-phenylethyl)amine NA 1000000 NA NA NA NA TTD
DPP4 1-Benzyl-N-(2-cyclopentylidene-2-fluoroethyl)-4-piperidinamine NA 250000 NA NA NA NA TTD
DPP4 (2-Cyclopentylidene-2-fluoroethyl)[3-(dimethylamino)propyl]amine NA 1000000 NA NA NA NA TTD
DPP4 N-(2-cyclohexylidene-2-fluoroethyl)cyclohexanamine NA 500000 NA NA NA NA TTD
DPP4 N-(2-cyclohexylidene-2-fluoroethyl)adamantan-1-amine NA 250000 NA NA NA NA TTD
DPP4 N-(2-cyclohexylidene-2-fluoroethyl)aniline NA 250000 NA NA NA NA TTD
DPP4 Benzyl(2-cyclohexylidene-2-fluoroethyl)amine NA 1000000 NA NA NA NA TTD
DPP4 (2-Cyclohexylidene-2-fluoroethyl)[(4-methoxyphenyl)methyl]amine NA 250000 NA NA NA NA TTD