| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| DPP4 |
[2-[Bis(2,2,2-trichloroethoxy)phosphoryl]pyrrolidin-1-yl]-pyrrolidin-2-ylmethanone;hydrochloride |
NA |
1800000 |
NA |
NA |
NA |
NA |
TTD |
| DPP4 |
[2-Bis(4-hydroxyphenoxy)phosphorylpyrrolidin-1-yl]-pyrrolidin-2-ylmethanone;hydrochloride |
NA |
190000 |
NA |
NA |
NA |
NA |
TTD |
| DPP4 |
Quercetin |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| DPP4 |
Rutin |
NA |
145000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| DPP4 |
Kaempferol |
NA |
132000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| DPP4 |
Baicalein |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| DPP4 |
3,7-Dihydroxyflavone |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| DPP4 |
1G244 |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP4 |
Baicalin |
NA |
225000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| DPP4 |
Talabostat |
NA |
21000000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP4 |
Ubenimex |
NA |
324300 |
NA |
NA |
NA |
NA |
PubChem |
| DPP4 |
2-(2,6-dimethylphenyl)-4-nitro-1H-isoindole-1,3(2H)-dione |
NA |
337500 |
NA |
NA |
NA |
NA |
TTD |
| DPP4 |
H-Val-Pro-Asp-Pro-Arg-NH2 |
142000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP4 |
ethyl 5,7-dihydroxy-2-(4-hydroxyphenyl)-3,4-dihydro-2H-chromene-8-carboxylate |
NA |
113760 |
NA |
NA |
NA |
NA |
TTD |
| DPP4 |
(2S)-1-[(2S)-2-amino-3-(furan-3-yl)propanoyl]pyrrolidine-2-carbonitrile |
NA |
113600 |
NA |
NA |
NA |
NA |
TTD |
| DPP4 |
2-{2-[Bis-(4-hydroxy-phenoxy)-phosphoryl]-pyrrolidine-1-carbonyl}-pyrrolidinium; chloride |
NA |
190000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP4 |
2-{2-[Bis-(2,2,2-trifluoro-ethoxy)-phosphoryl]-pyrrolidine-1-carbonyl}-pyrrolidinium; chloride |
NA |
9100000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP4 |
2-{2-[Bis-(2,2,2-trichloro-ethoxy)-phosphoryl]-pyrrolidine-1-carbonyl}-pyrrolidinium; chloride |
NA |
1800000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP4 |
2-(S)-Amino-4-benzylamino-1-piperidin-1-yl-butan-1-one |
NA |
247000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP4 |
3-Amino-4-oxo-4-pyrrolidin-1-yl-butyramide |
NA |
188000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |