| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| DPP4 |
(3S)-4-oxo-4-piperidin-1-ylbutane-1,3-diamine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| DPP4 |
D-Val-L-boroPro |
NA |
116000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP4 |
3-Amino-4-oxo-4-pyrrolidin-1-yl-butyric acid |
NA |
122000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP4 |
(S)-2,4-Diamino-1-piperidin-1-yl-butane-1-thione |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| DPP7 |
(R)-2,4-Diamino-1-piperidin-1-yl-butan-1-one |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP7 |
2-Amino-3-methyl-1-pyrrolidin-1-yl-pentan-1-one |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP7 |
N-[[(2S,3aS,7aS)-1-[(3R)-3-amino-4-(2,4,5-trifluorophenyl)butanoyl]-2,3,3a,4,5,6,7,7a-octahydroindol-2-yl]methyl]-1,1,1-trifluoromethanesulfonamide |
NA |
207350 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP7 |
N-Cyclohexyl-2-oxo-2-(1-piperidinyl)ethaneamine |
NA |
177000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP7 |
(2S)-2,6-diamino-1-(2-diphenoxyphosphorylpyrrolidin-1-yl)hexan-1-one |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| DPP7 |
(2-diphenoxyphosphorylpyrrolidin-1-yl)-[(2S)-pyrrolidin-2-yl]methanone |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| DPP7 |
diphenyl 1-((2S,3S)-2-amino-3-methylpentanoyl)pyrrolidin-2-ylphosphonate |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| DPP7 |
benzyl (S)-6-amino-1-(2-(diphenoxyphosphoryl)pyrrolidin-1-yl)-1-oxohexan-2-ylcarbamate |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| DPP7 |
Bis(4-acetamidophenyl) 1-(pyrrolidine-2-carbonyl)pyrrolidin-2-ylphosphonate |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| DPP7 |
(2S)-2-amino-1-(2-diphenoxyphosphorylpyrrolidin-1-yl)-3-phenyl-propan-1-one |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| DPP7 |
(2S,3S)-2-amino-1-(3-fluoropyrrolidin-1-yl)-3-methylpentan-1-one |
NA |
111000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP7 |
(2S,3S)-2-amino-1-(azetidin-1-yl)-3-methylpentan-1-one |
NA |
730000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP7 |
(2S,3S)-2-amino-1-(azepan-1-yl)-3-methylpentan-1-one |
NA |
228000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP7 |
(2S,3S)-2-amino-3-methyl-1-(2H-pyrrol-1(5H)-yl)pentan-1-one |
NA |
288000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP7 |
(2S,3S)-2-amino-1-(3-hydroxypyrrolidin-1-yl)-3-methylpentan-1-one |
NA |
299000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP7 |
(2S)-2-amino-N-(1-diphenoxyphosphorylethyl)butanediamide |
NA |
286000 |
NA |
NA |
NA |
NA |
BindingDB |