| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| DPP7 |
(S)-pyrrolidin-1-yl(pyrrolidin-2-yl)methanone |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| DPP7 |
US11096924, DASH-inhibitors 5320 |
NA |
53940000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP7 |
Xeruborbactam |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem |
| DPP7 |
US11096924, DASH-inhibitors 5349 |
NA |
610000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP7 |
US11096924, DASH-inhibitors 5363 |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP7 |
US11096924, DASH-inhibitors 5317 |
NA |
22060000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP7 |
US11096924, DASH-inhibitors 5553 |
NA |
978000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP7 |
US11096924, DASH-inhibitors 5311 |
NA |
63820000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP7 |
US11096924, DASH-inhibitors 5316 |
NA |
92160000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP7 |
US11096924, DASH-inhibitors 5325 |
NA |
842000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP7 |
US11096924, DASH-inhibitors 5554 |
NA |
36490000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP7 |
US11096924, DASH-inhibitors 4312 S |
NA |
610000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP7 |
(S)-benzyl 5-amino-6-(3,4-dihydroquinolin-1(2H)-yl)-6-oxohexylcarbamate |
NA |
390000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP7 |
US11096924, DASH-inhibitors 5322 |
NA |
36840000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP7 |
US11096924, DASH-inhibitors 5298 |
NA |
4180000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP7 |
US11096924, DASH-inhibitors 5333 |
NA |
26480000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP7 |
US11096924, DASH-inhibitors 5321 |
NA |
44850000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP7 |
US11096924, DASH-inhibitors 4312 |
NA |
6400000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP7 |
2-Amino-3-methyl-pentanoic acid diethylamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| DPP7 |
(S)-2-amino-4-methyl-1-(pyrrolidin-1-yl)pentan-1-one |
NA |
122000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |