| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| DPP7 |
2-Amino-3-methyl-pentanoic acid ethyl-methyl-amide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| DPP7 |
N-(2-cyclohexylidene-2-fluoroethyl)cyclohexanamine |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP7 |
N-(2-cyclohexylideneethyl)cyclohexanamine |
NA |
136000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP7 |
1-((2S,4S)-2-(2-tert-butyl-1,3,4-oxadiazole-5-carbonyl)-4-fluoropyrrolidin-1-yl)-2-(1-hydroxy-2-methylpropan-2-ylamino)ethanone |
NA |
145800 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP7 |
diphenyl 2-((2S,3R)-2-amino-3-methylpentanoyl)isoindolin-1-ylphosphonate |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| DPP7 |
di-(4-acetamido)phenyl 2-((S)-2,6-diaminohexanoyl)isoindolin-1-ylphosphonate |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| DPP7 |
di-(4-acetamido)phenyl 2-((2S,3S)-2-amino-3-methylpentanoyl)isoindolin-1-ylphosphonate |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| DPP7 |
diphenyl 2-((2S,3S)-2-amino-3-methylpentanoyl)isoindolin-1-ylphosphonate |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| DPP7 |
N-Cyclopentyl L-isoleucinamide |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP7 |
2-Amino-1-azepan-1-yl-3-methyl-pentan-1-one |
NA |
228000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP7 |
2-amino-N,N,3-trimethylpentanamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| DPP7 |
(2S,3R)-2-amino-1-(5-fluoroisoindolin-2-yl)-3-methylpentan-1-one |
NA |
30000000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP7 |
2,4-Diamino-1-piperidin-1-yl-butan-1-one |
NA |
191000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP7 |
N-(2-pyrrolidin-1-ylethyl)cyclohexanamine |
NA |
136000 |
NA |
NA |
NA |
NA |
TTD |
| DPP7 |
2-Amino-3-methyl-pentanoic acid methyl-propyl-amide |
NA |
213000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP7 |
Sitagliptin |
NA |
207350|654430 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| DPP7 |
2-Amino-3-(4-hydroxy-phenyl)-1-pyrrolidin-1-yl-propan-1-one |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP7 |
Ala-Pro-CN |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP7 |
Pyrrolidin-2-yl-pyrrolidin-1-yl-methanethione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| DPP7 |
2-Amino-1-(3-fluoro-pyrrolidin-1-yl)-3-methyl-pentan-1-one |
NA |
111000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |