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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
DPP7 (2S)-2-amino-N-(1-diphenoxyphosphorylpropyl)-3-methyl-pentanamide NA 1000000 NA NA NA NA BindingDB
DPP7 (2S)-2-amino-N-(1-diphenoxyphosphorylbutyl)-3-methyl-pentanamide NA 1000000 NA NA NA NA BindingDB
DPP7 (2S)-2-amino-N-(1-diphenoxyphosphoryl-2-methyl-propyl)-3-methyl-pentanamide NA 1000000 NA NA NA NA BindingDB
DPP7 (2S)-2-amino-N-(1-diphenoxyphosphoryl-2-methyl-butyl)-3-methyl-pentanamide NA 414000 NA NA NA NA BindingDB
DPP7 (2S)-2-amino-N-(1-diphenoxyphosphoryl-3-methyl-butyl)-3-methyl-pentanamide NA 286000 NA NA NA NA BindingDB
DPP7 (2S)-2-amino-N-[cyclohexyl(diphenoxyphosphoryl)methyl]-3-methyl-pentanamide NA 148000 NA NA NA NA BindingDB
DPP7 (2S)-2-amino-N-(2-cyclopenta-2,4-dien-1-yl-1-diphenoxyphosphoryl-ethyl)-3-methyl-pentanamide NA 288000 NA NA NA NA BindingDB
DPP7 (2S)-2-amino-N-[(4-cyanophenyl)-diphenoxyphosphoryl-methyl]-3-methyl-pentanamide NA 150000 NA NA NA NA BindingDB
DPP7 (2S)-2-amino-N-[(3-cyanophenyl)-diphenoxyphosphoryl-methyl]-3-methyl-pentanamide NA 509000 NA NA NA NA BindingDB
DPP7 N-[diphenoxyphosphoryl(phenyl)methyl]-2-(sec-butylamino)acetamide NA 109000 NA NA NA NA BindingDB
DPP7 (2S)-1-[(2S)-2-amino-3-(2-fluorophenyl)propanoyl]pyrrolidine-2-carbonitrile NA 296900 NA NA NA NA TTD
DPP7 (2S,4S)-1-[(2S)-2-amino-3-[2-(trifluoromethyl)phenyl]propanoyl]-4-fluoropyrrolidine-2-carbonitrile NA 102000 NA NA NA NA TTD
DPP7 Glu-boroSar NA 1700000 NA NA NA NA BindingDB
DPP7 Pyrrolidine, 1-[(2S,3R)-2-amino-3-methyl-1-oxopentyl]- NA 145000 NA NA NA NA BindingDB|TTD
DPP7 Nvp-dpp728 NA 110000|190000 NA NA NA NA BindingDB
DPP7 (2S,3S)-2-amino-3-methyl-1-(pyrrolidin-1-yl)pentan-1-one NA 110000 NA NA NA NA BindingDB
DPP7 3-Amino-4-oxo-4-pyrrolidin-1-yl-butyramide NA 152000 NA NA NA NA BindingDB|TTD
DPP7 2-Amino-1-(pyrrolidin-1-yl)propan-1-one NA 179000 NA NA NA NA BindingDB
DPP7 (S)-4-amino-5-oxo-5-(pyrrolidin-1-yl)pentanoic acid NA 1000000 NA NA NA NA TTD
DPP7 2-Amino-1-azetidin-1-yl-3-methyl-pentan-1-one NA 730000 NA NA NA NA BindingDB|TTD