| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| DPP8 |
(S)-2-amino-1-(pyrrolidin-1-yl)propan-1-one |
NA |
411000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP8 |
PT-630 |
NA |
33000000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP8 |
(2S)-2-amino-1-(2-diphenoxyphosphorylpyrrolidin-1-yl)-3-hydroxy-propan-1-one |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| DPP8 |
(2S)-2-amino-1-(2-diphenoxyphosphorylpyrrolidin-1-yl)-3-methyl-butan-1-one |
NA |
126000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP8 |
US11096924, DASH-inhibitors 5320 |
NA |
280000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP8 |
Xeruborbactam |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem |
| DPP8 |
US11096924, DASH-inhibitors 5349 |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP8 |
US11096924, DASH-inhibitors 5362 |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP8 |
US11096924, DASH-inhibitors 3102 A |
NA |
1200000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP8 |
US11096924, DASH-inhibitors 5363 |
NA |
270000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP8 |
2-[[2-[(3R)-3-aminopiperidin-1-yl]-4-oxo-5H-pyrrolo[3,2-d]pyrimidin-3-yl]methyl]-4-fluorobenzonitrile |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| DPP8 |
US11096924, DASH-inhibitors 5317 |
NA |
127500 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP8 |
US11096924, DASH-inhibitors 5311 |
NA |
80990000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP8 |
US11096924, DASH-inhibitors 5316 |
NA |
4112000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP8 |
US11096924, DASH-inhibitors 5325 |
NA |
123000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP8 |
US11096924, DASH-inhibitors 5323 |
NA |
862000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP8 |
(S)-benzyl 5-amino-6-(3,4-dihydroquinolin-1(2H)-yl)-6-oxohexylcarbamate |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| DPP8 |
US11096924, DASH-inhibitors 5322 |
NA |
2000000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP8 |
US11096924, DASH-inhibitors 5333 |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP8 |
US11096924, DASH-inhibitors 4160 |
NA |
400000|1400000 |
NA |
NA |
NA |
NA |
BindingDB |