| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| DPP8 |
(S)-1-((3R,4R)-3-amino-1-(1-(4-cyanophenyl)ethyl)pyrrolidine-4-carbonyl)pyrrolidine-2-carbonitrile |
NA |
1040000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP8 |
(1R,3S)-2-((3R,4R)-1-(4-(5-methyl-1,3,4-oxadiazol-2-yl)benzyl)-3-aminopyrrolidine-4-carbonyl)-3-fluorocyclopentanecarbonitrile |
NA |
332000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP8 |
4-(((3R,4R)-3-amino-4-((2R)-2-cyanocyclopentanecarbonyl)pyrrolidin-1-yl)methyl)-2,6-dimethylbenzonitrile |
NA |
346000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP8 |
4-(((3R,4R)-3-amino-4-((2R)-2-cyanocyclopentanecarbonyl)pyrrolidin-1-yl)methyl)-2,6-diethylbenzonitrile |
NA |
417000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP8 |
(1R)-2-((3R,4R)-1-(2-methyl-4-(1H-1,2,4-triazol-1-yl)benzyl)-3-aminopyrrolidine-4-carbonyl)cyclopentanecarbonitrile |
NA |
203000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP8 |
(S)-2,6-diamino-1-(3,4-dihydroquinolin-1(2H)-yl)hexan-1-one |
NA |
312000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP8 |
5-(aminomethyl)-N-cyclopropyl-4-(4-fluorophenyl)-6-methylpicolinamide |
106000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP8 |
(5-(Aminomethyl)-4-(4-fluorophenyl)-6-methylpyridin-2-yl)(pyrrolidin-1-yl)methanone |
137000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP8 |
5-(aminomethyl)-4-(2,4-difluorophenyl)-6-methyl-N-(5-methylisoxazol-3-yl)picolinamide |
179000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP8 |
5-(aminomethyl)-N-cyclopropyl-4-(2,4-difluorophenyl)-6-methylpicolinamide |
182000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP8 |
1G244 |
NA |
400000|1400000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP8 |
Ala-boroPro thioxoamide |
NA |
135000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP8 |
Talabostat |
NA |
5200000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP8 |
Pyrrolidine, 1-(N-phenylalanyl)- |
NA |
115000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP8 |
Glu-boroSar |
NA |
12000000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP8 |
(2S)-1-[(2S)-2-amino-3-(furan-3-yl)propanoyl]pyrrolidine-2-carbonitrile |
NA |
288200 |
NA |
NA |
NA |
NA |
TTD |
| DPP8 |
(2S)-1-[(2S)-2-amino-3-pyridin-2-ylpropanoyl]pyrrolidine-2-carbonitrile |
NA |
125100 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP8 |
(S)-4-amino-5-oxo-5-(pyrrolidin-1-yl)pentanoic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| DPP9 |
Ala-boroPro |
NA |
360000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP9 |
2-Oxo-2-pyrrolidin-1-ylethanamine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |