| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| DRD1 |
Cefepime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| DRD1 |
Ceftazidime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| DRD1 |
Tyramine |
390000 |
NA |
NA |
NA |
NA |
NA |
PubChem|TTD |
| DRD1 |
Aztreonam |
NA |
NA |
NA |
NA |
NA |
400000 |
PubChem |
| DRD1 |
Carumonam |
NA |
NA |
NA |
NA |
NA |
500000 |
PubChem |
| DRD1 |
Doripenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| DRD2 |
Imipenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| DRD2 |
2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine |
720000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DRD2 |
1-(2-Methoxyphenyl)-6-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-1,6-diazaspiro[3.3]heptane |
114945 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DRD2 |
3-(4-Methoxyphenyl)-9-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-3,9-diazaspiro[5.5]undecane |
104847 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DRD2 |
1-(4-Fluorophenyl)-6-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-1,6-diazaspiro[3.3]heptane |
109574 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DRD2 |
[4-[2-[Bis(4-fluorophenyl)methylsulfinyl]ethylamino]piperidin-1-yl]-(4-fluorophenyl)methanone |
156000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| DRD2 |
3-[3-[(4-Methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-3,9-diazaspiro[5.5]undecane |
225748 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DRD2 |
6,9-Dichloro-3-methyl-1-phenyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine-7,8-diol; hydrochloride |
810000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DRD2 |
5-Chloro-2-[3-(4-pyridin-2-ylpiperazin-1-yl)propyl]-1,3-benzothiazole |
NA |
NA |
NA |
1800000 |
NA |
NA |
BindingDB |
| DRD2 |
D4R agonist-1 |
NA |
NA |
NA |
936000 |
NA |
NA |
BindingDB |
| DRD2 |
6-Methyl-2-[3-(4-pyridin-2-ylpiperidin-1-yl)propyl]-1,3-benzothiazole |
NA |
NA |
NA |
496000 |
NA |
NA |
BindingDB |
| DRD2 |
2-[4-(4-Pyridin-2-ylpiperazin-1-yl)butyl]-1,3-benzothiazole |
NA |
NA |
NA |
124000 |
NA |
NA |
BindingDB |
| DRD2 |
7-Methoxy-2-[3-(4-pyridin-2-ylpiperidin-1-yl)propyl]-1,3-benzothiazole |
NA |
NA |
NA |
183000 |
NA |
NA |
BindingDB |
| DRD2 |
4-Chloro-2-[3-(4-pyridin-2-ylpiperazin-1-yl)propyl]-1,3-benzothiazole |
NA |
NA |
NA |
2052000 |
NA |
NA |
BindingDB |