| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| DRD2 |
6-Chloro-2-[3-(4-pyridin-2-ylpiperazin-1-yl)propyl]-1,3-benzothiazole |
NA |
NA |
NA |
1620000 |
NA |
NA |
BindingDB |
| DRD2 |
6-Methyl-2-[3-(4-pyridin-2-ylpiperazin-1-yl)propyl]-1,3-benzothiazole |
NA |
NA |
NA |
591000 |
NA |
NA |
BindingDB |
| DRD2 |
6-Methoxy-2-[3-(4-pyridin-2-ylpiperidin-1-yl)propyl]-1,3-benzothiazole |
NA |
NA |
NA |
228000 |
NA |
NA |
BindingDB |
| DRD2 |
1-Phenyl-2,3,4,9-tetrahydro-1H-beta-carboline |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DRD2 |
3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-4-(3''-chlorophenyl)piperazine |
298000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DRD2 |
5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}pentyl-4-(3''-chlorophenyl)piperazine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DRD2 |
3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-4-(3''-trifluoromethylphenyl)piperazine |
1412000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DRD2 |
2{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-4-(2''-methoxyphenyl)piperazine |
427000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DRD2 |
5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}pentyl-4-(2''-methoxyphenyl)piperazine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DRD2 |
3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-4-(4''-fluorophenyl)piperazine |
655000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DRD2 |
5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}pentyl-4-(4''-fluorophenyl)piperazine |
847000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DRD2 |
2-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-4-(2''-pyrimidil)piperazine |
629000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DRD2 |
4-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-4-(2''-pyrimidyl)piperazine |
854000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DRD2 |
3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-4-(3''-methyl)piperazine |
565000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DRD2 |
5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}pentyl-4-(N-methyl)piperazine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DRD2 |
3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-(3,4-dihydroisoquinoline) |
114000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DRD2 |
4{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-(3,4-dihydroisoquinoline) |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DRD2 |
2-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-(6,7-dimethoxy-3,4-dihydroisoquinoline) |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DRD2 |
4-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-(6,7-dimethoxy-3,4-dihydroisoquinoline) |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DRD2 |
2-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-4-(3''-chlorophenyl)piperazine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |