| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| DRD2 |
4{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-4-(3''-trifluoromethylphenyl)piperazine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DRD2 |
4{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-4-(4''-fluorophenyl)piperazine |
1324000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DRD2 |
2-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-4-(N-methyl)piperazine |
178000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DRD2 |
4-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-4-(N-methyl)piperazine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DRD2 |
2-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-(3,4-dihydroisoquinoline) |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DRD2 |
5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}pentyl-(3,4-dihydroisoquinoline) |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DRD2 |
3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-(6,7-dimethoxy-3,4-dihydroisoquinoline) |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DRD2 |
5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-(6,7-dimethoxy-3,4-dihydroisoquinoline) |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DRD2 |
5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}pentyl-4-(2''-pyrimidyl)piperazine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DRD2 |
4-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-4-(3''-trifluoromethylphenyl)piperazine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DRD2 |
2-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-4-(3''-trifluoromethyl)piperazine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DRD2 |
2{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-4-(4''-fluorophenyl)piperazine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DRD2 |
4-Methyl-3-phenyl-5-propylsulfanyl-1,2,4-triazole |
180375 |
NA |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| DRD2 |
Cefazolin |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| DRD2 |
Meropenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| DRD2 |
6-methoxy-1-(1-methyl-4-nitro-1H-pyrrol-2-yl)-4,9-dihydro-3H-pyrido[3,4-b]indole |
200000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DRD2 |
(E)-6-((3,4-dihydroisoquinolin-2(1H)-yl)methyleneamino)-2,3-dihydro-1H-inden-1-ol |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DRD2 |
(4aS,5R,10bR)-5-phenyl-1,2,3,4,4a,5,6,10b-octahydrobenzo[h]isoquinoline-7,8-diol |
750000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| DRD2 |
Cefepime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| DRD2 |
Ceftazidime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |