Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| DRD2 | Tyramine | 160000 | NA | NA | NA | NA | NA | BindingDB|PubChem |
| DRD2 | 2-[3-(4-Pyrimidin-2-ylpiperazin-1-yl)propyl]-1,3-benzothiazole | NA | NA | NA | 1180000 | NA | NA | BindingDB |
| DRD2 | Aztreonam | NA | NA | NA | NA | NA | 400000 | PubChem |
| DRD2 | Carumonam | NA | NA | NA | NA | NA | 500000 | PubChem |
| DRD2 | Doripenem | NA | NA | NA | NA | NA | 300000 | PubChem |
| DRD2 | 4-(3-Chlorophenyl)piperazine-1-carboxamide | 115900 | NA | NA | NA | NA | NA | BindingDB |
| DRD2 | N-Acetyldeclopramide | NA | 975000 | NA | NA | NA | NA | BindingDB |
| DRD2 | (E)-6-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)methyleneamino)-2,3-dihydro-1H-inden-1-ol | 300000 | NA | NA | NA | NA | NA | TTD |
| DRD3 | Imipenem | NA | NA | NA | NA | NA | 300000 | PubChem |
| DRD3 | 1-(4-Fluorophenyl)-6-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]-1,6-diazaspiro[3.3]heptane | 181888 | NA | NA | NA | NA | NA | TTD |
| DRD3 | 6-Methyl-2-[3-(4-pyridin-2-ylpiperazin-1-yl)propyl]-1,3-benzothiazole | 201000 | NA | NA | NA | NA | NA | BindingDB |
| DRD3 | Cefazolin | NA | NA | NA | NA | NA | 300000 | PubChem |
| DRD3 | Fenofibrate | NA | 137533 | NA | NA | NA | NA | PubChem |
| DRD3 | Meropenem | NA | NA | NA | NA | NA | 300000 | PubChem |
| DRD3 | Cefepime | NA | NA | NA | NA | NA | 300000 | PubChem |
| DRD3 | Ceftazidime | NA | NA | NA | NA | NA | 300000 | PubChem |
| DRD3 | Aztreonam | NA | NA | NA | NA | NA | 400000 | PubChem |
| DRD3 | Carumonam | NA | NA | NA | NA | NA | 500000 | PubChem |
| DRD3 | Doripenem | NA | NA | NA | NA | NA | 300000 | PubChem |
| DRD4 | (4aS,5R,10bR)-5-phenyl-1,2,3,4,4a,5,6,10b-octahydrobenzo[h]isoquinoline-7,8-diol | 2650000 | NA | NA | NA | NA | NA | BindingDB|TTD |