| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| DUSP10 |
[[3-(3-Cyclohexyl-2-oxidanyl-phenyl)phenyl]-bis(fluoranyl)methyl]phosphonic acid |
150000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUSP22 |
5-{4-Oxo-5-[1-phenyl-meth-(Z)-ylidene]-2-thioxo-thiazolidin-3-yl}-isophthalic acid |
NA |
103000 |
NA |
NA |
NA |
NA |
BindingDB |
| DUSP22 |
3-{5-[1-(4-Hydroxy-phenyl)-meth-(Z)-ylidene]-4-oxo-2-thioxo-thiazolidin-3-yl}-benzoic acid |
NA |
157000 |
NA |
NA |
NA |
NA |
BindingDB |
| DUSP3 |
2-(4-(7-(4-Methoxybenzoyl)cyclopenta[d][1,2]oxazin-4-yl)phenoxy)acetic acid |
NA |
181200 |
NA |
NA |
NA |
NA |
BindingDB |
| DUSP3 |
4-(5-((3-Carboxy-4-hydroxyphenyl)amino)-5-oxopentanamido)-2,2,6,6-tetramethylpiperidin-1-olate |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| DUSP3 |
2-Hydroxy-5-(5-(((1-hydroxy-2,2,6,6-tetramethylpiperidin-4-yl)amino)methyl)furan-2-yl)benzoic acid |
NA |
241000 |
NA |
NA |
NA |
NA |
BindingDB |
| DUSP3 |
(E)-2,2,6,6-tetramethyl-4-(3-(5-(3-nitrophenyl)furan-2-yl)acrylamido)piperidin-1-olate |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| DUSP3 |
(E)-2,2,6,6-tetramethyl-4-(3-(5-(4-nitrophenyl)furan-2-yl)acrylamido)piperidin-1-olate |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| DUSP3 |
Methyl 2-hydroxy-5-(5-(((1-hydroxy-2,2,6,6-tetramethylpiperidin-4-yl)amino)methyl)furan-2-yl)benzoate |
NA |
850000 |
NA |
NA |
NA |
NA |
BindingDB |
| DUSP3 |
4-[2-[[3,5-Bis[3-[4-[difluoro(phosphono)methyl]phenyl]propanoylamino]benzoyl]amino]ethyl]benzoic acid |
3600000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| DUSP3 |
6-hydroxy-3-(1-(4-(naphthalen-1-ylamino)-4-oxobutyl)-1H-1,2,3-triazol-4-yl)-2-phenylbenzofuran-5-carboxylic acid |
NA |
103000 |
NA |
NA |
NA |
NA |
BindingDB |
| DUSP3 |
2-Hydroxy-5-{4-oxo-5-[1-phenyl-meth-(Z)-ylidene]-2-thioxo-thiazolidin-3-yl}-benzoic acid |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB |
| DUSP3 |
1-((1S,4aS,8aS)-2,5,5,8a-Tetramethyl-1,4,4a,5,6,7,8,8a-octahydro-naphthalen-1-yl)-pent-4-en-2-ol |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB |
| DUSP3 |
2-[(1S,4aS,8aS)-2,5,5,8a-tetramethyl-1,4,4a,6,7,8-hexahydronaphthalen-1-yl]ethyl hydrogen sulfate |
NA |
275000 |
NA |
NA |
NA |
NA |
BindingDB |
| DUSP3 |
Hydrogen (2-naphthyloxy)methylphosphonate |
5700000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| DUSP3 |
Dioxido-oxo-(phenoxymethyl)-lambda5-phosphane |
26000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| DUSP3 |
[4-(4-Hydroxybenzyl)phenoxy]methylphosphonate |
1300000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| DUSP3 |
Hydrogen (1-phenanthryloxy)methylphosphonate |
570000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| DUSP3 |
Hydrogen (1-naphthyloxy)methylphosphonate |
4800000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| DUSP3 |
[4-(Carboxymethyl)phenoxy]methylphosphonate |
2600000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |