| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| DUT |
1-(6-Tritylaminohexyl)uracil |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
1-(3-Trityloxypropyl)pyrimidine-2,4-dione |
313000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DUT |
1-(5-Trityloxypentyl)uracil |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
1-[2-(Hydroxymethyl)-4-(trityloxy)butyl]uracil |
260000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DUT |
1-(3-Hydroxypropyl)uracil |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
1-[2-(Benzoyloxyethoxy)methyl]uracil |
311000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DUT |
1-(6-Benzoyloxyhexyl)uracil |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
1-(4-Tritylaminobutyl)uracil |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
1-(5-Tritylaminopentyl)uracil |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
{3-[(tert-butyldimethylsilyl)oxy]-5-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)oxolan-2-yl}methyl N-sulfamoylcarbamate |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
Phosphoric acid 3-(tert-butyl-dimethyl-silanyloxy)-5-(2,4-dioxo-3,4-dihydro-2H-pyrimidin-1-yl)-tetrahydro-furan-2-ylmethyl ester diethyl ester |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
1-(4-Tert-butyldiphenylsilyloxyhexyl)uracil |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
(Diethoxy-phosphoryl)-acetic acid 5-(2,4-dioxo-3,4-dihydro-2H-pyrimidin-1-yl)-3-hydroxy-tetrahydro-furan-2-ylmethyl ester |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
Sulfamic acid 5-(2,4-dioxo-3,4-dihydro-2H-pyrimidin-1-yl)-3-hydroxy-tetrahydro-furan-2-ylmethyl ester |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
1-[4-(tert-Butyl-dimethyl-silanyloxy)-5-trityloxymethyl-tetrahydro-furan-2-yl]-1H-pyrimidine-2,4-dione |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
1-(6-Triphenylsilyloxyhexyl)uracil |
383000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DUT |
Pentanoic acid 5-(2,4-dioxo-3,4-dihydro-2H-pyrimidin-1-yl)-3-hydroxy-tetrahydro-furan-2-ylmethyl ester |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
[(2R,3S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3-hydroxyoxolan-2-yl]methyl diphenyl phosphate |
135000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DUT |
[(2R,3S,5R)-3-[tert-butyl(dimethyl)silyl]oxy-5-(2,4-dioxopyrimidin-1-yl)oxolan-2-yl]methyl diphenyl phosphate |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
1-[4-(Tert-butoxycarbonylamino)-3-(trityloxymethyl)butyl]- |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |