| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| DUT |
N-[4-(tert-butyl diphenyl silanyloxy)-butyl]-2-uracil acetamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
1-[N-(3-triphenylmethylaminopropyl)-acetamide] uracil |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
1-[N-(triphenylmethylaminoethyl)-N-(aminoethyl) acetamide] uracil |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
1-[N-(triphenylmethyl) diaminodi (n-propyl) acetamide] uracil |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
1-(5-Aminomethyl-4-hydroxy-tetrahydro-furan-2-yl)-1H-pyrimidine-2,4-dione |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
Acetic acid 5-(2,4-dioxo-3,4-dihydro-2H-pyrimidin-1-yl)-3-hydroxy-tetrahydro-furan-2-ylmethyl ester |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
1-{(2S,5S)-4-Fluoro-5-[(trityloxy)methyl]tetrahydrofuran-2-YL}pyrimidine-2,4(1H,3H)-dione |
457000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DUT |
dUTPase inhibitor, 1 |
135000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| DUT |
dUTPase inhibitor, 6 |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
dUTPase inhibitor, 7 |
807000|808000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DUT |
1-(4-Fluoro-5-triphenylsilanyloxymethyl-tetrahydro-furan-2-yl)-1H-pyrimidine-2,4-dione |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
1-{4-(tert-Butyl-dimethyl-silanyloxy)-5-[(trityl-amino)-methyl]-tetrahydro-furan-2-yl}-1H-pyrimidine-2,4-dione |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
1-[4-[Tert-butyl(dimethyl)silyl]oxy-5-[(diphenoxyphosphorylamino)methyl]oxolan-2-yl]pyrimidine-2,4-dione |
232000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DUT |
1-(4-Hydroxy-5-triisopropylsilanyloxymethyl-tetrahydro-furan-2-yl)-1H-pyrimidine-2,4-dione |
1000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| DUT |
dUTPase inhibitor, 9 |
805000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| DUT |
1-(4-Hydroxy-5-triphenylsilanyloxymethyl-tetrahydro-furan-2-yl)-1H-pyrimidine-2,4-dione |
908000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| DUT |
1-[5-[(Diphenoxyphosphorylamino)methyl]-4-hydroxyoxolan-2-yl]pyrimidine-2,4-dione |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
2-diethoxyphosphoryl-N-[[5-(2,4-dioxopyrimidin-1-yl)-3-hydroxyoxolan-2-yl]methyl]acetamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
N-[[5-(2,4-dioxopyrimidin-1-yl)-3-hydroxyoxolan-2-yl]methyl]tricyclo[5.2.1.03,8]decane-1-carboxamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
N-[5-(2,4-Dioxo-3,4-dihydro-2H-pyrimidin-1-yl)-3-hydroxy-tetrahydro-furan-2-ylmethyl]-acetamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |