| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| DUT |
2',3'-Didehydro-2',3'-dideoxyuridine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
5'-O-Triisopropylsilyl-2'-deoxyuridine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
Triphenylsilanol |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
N-[3-(3-benzoyl-2,4-dioxo-pyrimidin-1-yl)propyl]-2,2,2-triphenyl-acetamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DUT |
N-[3-(2,4-dioxopyrimidin-1-yl)propyl]-2,2-diphenyl-acetamide |
286000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DUT |
N-[3-(2,4-dioxopyrimidin-1-yl)propyl]-2,2,2-triphenyl-acetamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DUT |
4-(2,4-dioxopyrimidin-1-yl)-N-trityl-butanamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DUT |
N-(3-hydroxypropyl)-2,2,2-triphenyl-acetamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DVL1 |
2-(2-Methoxy-4-{[(2Z)-3-oxo-2,3-dihydro-1-benzothiophen-2-ylidene]methyl}phenoxy)acetic acid |
NA |
NA |
268000 |
NA |
NA |
NA |
BindingDB |
| DVL1 |
1-[2-(5-Chlorothiophen-2-yl)quinoline-4-carbonyl]piperidine-4-carboxylic acid |
NA |
NA |
311000 |
NA |
NA |
NA |
BindingDB |
| DVL1 |
6-methyl-2-(2-methylbutylcarbamoyl)-3-(2-phenylethyl)-1H-indole-5-carboxylic acid |
NA |
159000 |
NA |
NA |
NA |
NA |
BindingDB |
| DVL1 |
2-(benzylcarbamoyl)-6-methyl-3-(2-phenylethyl)-1H-indole-5-carboxylic acid |
NA |
197000 |
NA |
NA |
NA |
NA |
BindingDB |
| DVL1 |
2-(cyclohexylmethylcarbamoyl)-6-methyl-3-(2-phenylethyl)-1H-indole-5-carboxylic acid |
NA |
157000 |
NA |
NA |
NA |
NA |
BindingDB |
| DVL1 |
{2-chloro-4-[(Z)-(5-oxo-1-propyl-2-thioxoimidazolidin-4-ylidene)methyl]phenoxy}acetic acid |
NA |
NA |
152000 |
NA |
NA |
NA |
BindingDB |
| DVL1 |
2-[[3-[(2-phenylacetyl)amino]benzoyl]amino]benzoic Acid |
NA |
NA |
954000 |
NA |
NA |
NA |
BindingDB |
| DVL1 |
3-(5-{(E)-[3-(2-methoxy-2-oxoethyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl}furan-2-yl)-2-methylbenzoic acid |
NA |
NA |
251000 |
NA |
NA |
NA |
BindingDB |
| DVL1 |
methyl 2-[4-[(Z)-(3-oxo-1-benzothiophen-2-ylidene)methyl]phenoxy]acetate |
NA |
NA |
783000 |
NA |
NA |
NA |
BindingDB |
| DVL1 |
2-[6-(4-Chloro-2-fluorophenyl)sulfonyloxy-1-benzofuran-3-yl]acetic acid |
NA |
NA |
139000 |
NA |
NA |
NA |
BindingDB |
| DVL3 |
6-methyl-2-(2-methylbutylcarbamoyl)-3-(2-phenylethyl)-1H-indole-5-carboxylic acid |
NA |
160000 |
NA |
NA |
NA |
NA |
BindingDB |
| DVL3 |
2-(benzylcarbamoyl)-6-methyl-3-(2-phenylethyl)-1H-indole-5-carboxylic acid |
NA |
291000 |
NA |
NA |
NA |
NA |
BindingDB |