| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| EDNRA |
4-(1,1,1,3,3,3-hexafluoro-2-methoxypropan-2-yl)-N-[6-(2-hydroxyethoxy)-5-(2-methoxyphenoxy)-2-pyrimidin-2-ylpyrimidin-4-yl]benzenesulfonamide |
NA |
693000 |
NA |
NA |
NA |
NA |
TTD |
| EDNRA |
o-Deshydroxyethyl bosentan |
NA |
133000 |
NA |
NA |
NA |
NA |
TTD |
| EDNRA |
Moxifloxacin |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| EDNRA |
(8-Benzyloxy-11-oxo-5,11-dihydro-dibenzo[b,e][1,4]diazepin-10-yl)-acetic acid |
109000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| EDNRA |
(-)-(S)-9-Fluoro-2,3-dihydro-3-methyl-10-(4-methyl-1-piperazinyl)-7-oxo-7H-pyrido(1,2,3-de)-1,4-benzoxazine-6-carboxylic acid, hemihydrate |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| EDNRA |
Cefazolin |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| EDNRA |
Meropenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| EDNRA |
(2E,4E,6E)-Octa-2,4,6-trienoic acid (5R,9aS,9bS)-9b-hydroxy-6,6,9a-trimethyl-1-oxo-1,3,5,5a,6,7,8,9,9a,9b-decahydro-naphtho[1,2-c]furan-5-yl ester |
NA |
135000 |
NA |
NA |
NA |
NA |
TTD |
| EDNRA |
Ofloxacin |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| EDNRA |
Cefepime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| EDNRA |
Ceftazidime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| EDNRA |
Aztreonam |
NA |
NA |
NA |
NA |
NA |
400000 |
PubChem |
| EDNRA |
Carumonam |
NA |
NA |
NA |
NA |
NA |
500000 |
PubChem |
| EDNRA |
Doripenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| EDNRA |
4-[(2R,3R)-3-[(3,4-Dimethoxyphenyl)methyl]-4-methoxy-2-(methoxymethyl)butyl]-1,2-dimethoxybenzene |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| EDNRB |
(5S,6R,7R)-5-(3,4-dimethoxyphenyl)-4-methoxy-6,7-bis(methoxymethyl)-5,6,7,8-tetrahydrobenzo[f][1,3]benzodioxole |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| EDNRB |
4''-(2-Methyl-oxazol-4-yl)-biphenyl-2-sulfonic acid (3,4-dimethyl-isoxazol-5-yl)-amide |
110000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| EDNRB |
N-(4-bromo-3-methyl-5-isoxazolyl)-2-[N-(3-carboxyphenyl)aminocarbonyl]thiophene-3-sulfonamide |
NA |
117000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| EDNRB |
Hypophyllanthin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| EDNRB |
2,4-Dichloro-N-(3,4-dimethyl-isoxazol-5-yl)-benzenesulfonamide |
NA |
105000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |