| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| DVL3 |
2-(cyclohexylmethylcarbamoyl)-6-methyl-3-(2-phenylethyl)-1H-indole-5-carboxylic acid |
NA |
309000 |
NA |
NA |
NA |
NA |
BindingDB |
| DYRK1A |
3,4,5-Trimethylpyrazole |
NA |
NA |
215000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| DYRK1A |
CID 145986658 |
NA |
420000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DYRK1A |
5-Chloro-2-hydroxynicotinic acid |
NA |
NA |
680000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| DYRK1A |
5-(Benzylamino)pyrimido[4,5-c]quinoline-8-carboxylic acid |
NA |
760000 |
NA |
NA |
NA |
NA |
BindingDB |
| DYRK1A |
(6-Chloroimidazo(2,1-b)(1,3)thiazol-5-yl)methanol |
NA |
NA |
658000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| DYRK1A |
6-chloro-1H-indazole |
NA |
NA |
180000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| DYRK1A |
O6-(R)-Roscovitine, R-2-(6-benzyloxy-9-isopropyl-9H-purin-2-ylamino)-butan-1-OL |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB |
| DYRK1A |
6-Bromo-1H-1,2,3-triazolo[4,5-b]pyridine |
NA |
NA |
533000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| DYRK1A |
N-(4-methoxybenzyl)benzofuro[2,3-b]pyridin-4-amine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DYRK1A |
4-chloro-5H-pyrrolo[3,2-d]pyrimidine |
NA |
NA |
163000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| DYRK1A |
1H-Benzotriazol-6-amine |
NA |
NA |
430000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| DYRK2 |
AZ191 |
NA |
190000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ECE1 |
(2S)-2-[[(2S)-2-[[ethoxy(hydroxy)phosphoryl]amino]-4-methylpentanoyl]amino]-3-(1H-indol-3-yl)propanoic acid |
NA |
109000 |
NA |
NA |
NA |
NA |
TTD |
| ECE1 |
3-(Naphthalene-2-sulfonyl)-heptanoic acid hydroxyamide |
NA |
450000 |
NA |
NA |
NA |
NA |
TTD |
| ECE1 |
Xeruborbactam |
NA |
431000 |
NA |
NA |
NA |
NA |
PubChem |
| EDNRA |
(2S,4S)-5,8-dimethoxy-6-methyl-4-phenyl-1,2,3,4-tetrahydronaphthalene-2-carboxylic Acid |
NA |
160000 |
NA |
NA |
NA |
NA |
TTD |
| EDNRA |
Imipenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| EDNRA |
3-[[4-[2-[(3,4-dimethyl-1,2-oxazol-5-yl)sulfamoyl]phenyl]phenyl]methyl]-N-[2-(4-methoxyphenyl)ethyl]-7-methyl-2-propylbenzimidazole-5-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| EDNRA |
N-tert-butyl-3-[[4-[2-[(3,4-dimethyl-1,2-oxazol-5-yl)sulfamoyl]phenyl]phenyl]methyl]-7-methyl-2-propylbenzimidazole-5-carboxamide |
NA |
140000 |
NA |
NA |
NA |
NA |
TTD |