| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| EDNRB |
4''-Pyrimidin-4-yl-biphenyl-2-sulfonic acid (3,4-dimethyl-isoxazol-5-yl)-amide |
130000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| EDNRB |
4''-Pyrimidin-5-yl-biphenyl-2-sulfonic acid (3,4-dimethyl-isoxazol-5-yl)-amide |
170000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| EDNRB |
4''-(1H-Imidazol-2-yl)-biphenyl-2-sulfonic acid (3,4-dimethyl-isoxazol-5-yl)-amide |
150000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| EDNRB |
4''-(1-Methyl-1H-imidazol-2-yl)-biphenyl-2-sulfonic acid (3,4-dimethyl-isoxazol-5-yl)-amide |
120000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| EDNRB |
3-[(4-chloro-3-methyl-1,2-oxazol-5-yl)sulfamoyl]-N-(4-methyl-1,3-benzodioxol-5-yl)thiophene-2-carboxamide |
NA |
355500 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| EDNRB |
3-Benzo[1,3]dioxol-5-yl-5-ethoxy-1-(4-methoxy-benzyl)-1H-indole-2-carboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| EDNRB |
N-(3,4-dimethyl-1,2-oxazol-5-yl)-2-[4-(2H-tetrazol-5-yl)phenyl]benzenesulfonamide |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| EDNRB |
(2E,4E)-Hexa-2,4-dienoic acid (5R,9aS,9bS)-1,9b-dihydroxy-6,6,9a-trimethyl-1,3,5,5a,6,7,8,9,9a,9b-decahydro-naphtho[1,2-c]furan-5-yl ester |
NA |
148000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| EDNRB |
N-(3,4-Dimethyl-isoxazol-5-yl)-2-pyridin-3-yl-benzenesulfonamide |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| EDNRB |
N-(3,4-Dimethyl-isoxazol-5-yl)-2-(1H-indol-3-yl)-benzenesulfonamide |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| EDNRB |
N-(3,4-Dimethyl-isoxazol-5-yl)-2-pyrimidin-2-yl-benzenesulfonamide |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| EDNRB |
Acridin-9-yl-benzo[1,3]dioxol-5-yl-acetic acid methyl ester |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| EDNRB |
N-(3,4-Dimethyl-isoxazol-5-yl)-2-thiophen-3-yl-benzenesulfonamide |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| EDNRB |
N-(3,4-Dimethyl-isoxazol-5-yl)-2-thiophen-2-yl-benzenesulfonamide |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| EDNRB |
4-[(2R,3R)-3-[(3,4-Dimethoxyphenyl)methyl]-4-methoxy-2-(methoxymethyl)butyl]-1,2-dimethoxybenzene |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| EED |
3-Benzylpiperidine |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| EED |
3-(1-Benzofuran-7-ylmethyl)piperidine-1-carboxamide |
NA |
174000 |
NA |
NA |
NA |
NA |
TTD |
| EED |
3-((4-Methoxyphenyl)methyl)piperidine |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| EED |
3-(2-Methoxy-benzyl)-piperidine |
NA |
146000 |
NA |
NA |
NA |
NA |
TTD |
| EED |
3-[(4-Fluoro-3-methoxyphenyl)methyl]piperidine |
NA |
119000 |
NA |
NA |
NA |
NA |
TTD |