| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| DUT |
1-(4-Benzyloxycarbonylaminobutyl)uracil |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
Sulfamic acid 3-(tert-butyl-dimethyl-silanyloxy)-5-(2,4-dioxo-3,4-dihydro-2H-pyrimidin-1-yl)-tetrahydro-furan-2-ylmethyl ester |
324000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DUT |
1-(3-Benzoyloxypropyl)uracil |
898000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DUT |
1-(5-Triphenylsilyloxypentyl)uracil |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
1-[2-(Trityloxy)ethoxymethyl]uracil |
NA |
185000 |
NA |
NA |
NA |
NA |
BindingDB |
| DUT |
1-(4-Hydroxybutyl)uracil |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
US10858344, Example 91 |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB |
| DUT |
US10858344, Example 94 |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB |
| DUT |
5'-O-Benzoyl-2'-deoxyuridine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
1-(5-Trityloxymethyl-2,5-dihydro-furan-2-yl)-1H-pyrimidine-2,4-dione |
156000|157000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DUT |
dUTPase inhibitor, 5 |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
1-[(2R,5S)-5-[[tert-butyl(diphenyl)silyl]oxymethyl]-2,5-dihydrofuran-2-yl]pyrimidine-2,4-dione |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
1-((2R,4S,5R)-5-((tert-butyldiphenylsilyloxy)methyl)-4-hydroxytetrahydrofuran-2-yl)pyrimidine-2,4(1H,3H)-dione |
806000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DUT |
US10858344, Example 106 |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB |
| DUT |
N-(3-hydroxypropyl)-2,2-diphenyl-acetamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DUT |
4-(2,4-Dioxopyrimidin-1-yl)butanoic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DUT |
1-[N-hydroxyethyl-N-(triphenylmethyl amino) ethyl-acetamide] uracil |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
1-[N-(2-triphenylmethylaminoethyl)-acetamide] uracil |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
1-[N-(3-triphenylmethylaminobutyl)-acetamide] uracil |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
N-[3-(tert-butyl diphenyl silanyloxy)-propyl]-2-uracil acetamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |