| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| DUSP3 |
1-ethyl-6-methyl-3-[(E)-2-phenylethenyl]pyrimido[5,4-e][1,2,4]triazine-5,7-dione |
NA |
106000 |
NA |
NA |
NA |
NA |
BindingDB |
| DUSP3 |
3-[(5Z)-5-(4-methylbenzylidene)-4-oxo-2-thioxo-1,3-thiazolidin-3-yl]benzoic acid |
NA |
123000 |
NA |
NA |
NA |
NA |
BindingDB |
| DUSP3 |
Cefsulodin |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem |
| DUSP3 |
|
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB |
| DUSP3 |
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N'-[(5-{4-nitrophenyl}-2-furyl)methylene]-2-furohydrazide |
NA |
123000 |
NA |
NA |
NA |
NA |
BindingDB |
| DUSP3 |
|
NA |
158000 |
NA |
NA |
NA |
NA |
BindingDB |
| DUSP3 |
4-((S)-(S)-1-Carbamoyl-3-carboxy-propylcarbamoyl)-4-{2-[4-(3-oxo-propenyl)-benzoylamino]-acetylamino}-butyric acid |
290000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| DUSP3 |
4-{5-[(1,3-dioxo-1,3-dihydro-2H-inden-2-ylidene)methyl]furan-2-yl}-3-methylbenzoic acid |
NA |
147300 |
NA |
NA |
NA |
NA |
BindingDB |
| DUT |
1-[4-(tert-Butyl-dimethyl-silanyloxy)-5-hydroxymethyl-tetrahydro-furan-2-yl]-1H-pyrimidine-2,4-dione |
119000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DUT |
[(2R,3S,5R)-5-(2,4-dioxopyrimidin-1-yl)-3-hydroxyoxolan-2-yl]methyl diethyl phosphate |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
5'-O-(Dimethoxytrityl)-5-(propargyloxy)-2'-deoxyuridine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
5'O-trityl-2',3'-dideoxy-2',3'-didehydrouridine |
157000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DUT |
1-(4-Triphenylsilyloxybutyl)uracil |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
1-(4-Trityloxybutyl)uracil |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
({[5-(2,4-Dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-3-hydroxyoxolan-2-yl]methoxy}carbonyl)(sulfamoyl)azanide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
1-(6-Trityloxyhexyl)uracil |
476000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DUT |
1-(5-Hydroxypentyl)uracil |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
1-[2-(Azidomethyl)-4-(trityloxy)butyl]uracil |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
1-(4-Tert-butyloxycarbamatebutyl)uracil |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| DUT |
1-[(E)-4-trityloxy-2-butenyl]uracil |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |