Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| DPP9 | (2S,3aS,6aS)-1-[(3R)-3-amino-4-phenylbutanoyl]-3,3a,4,5,6,6a-hexahydro-2H-cyclopenta[b]pyrrole-2-carbonitrile | NA | 107660 | NA | NA | NA | NA | BindingDB|TTD |
| DPP9 | Xeruborbactam | NA | 1000000 | NA | NA | NA | NA | PubChem |
| DPP9 | US11096924, DASH-inhibitors 5349 | NA | 3100000 | NA | NA | NA | NA | BindingDB |
| DPP9 | 2-[[2-[(3R)-3-aminopiperidin-1-yl]-4-oxo-5H-pyrrolo[3,2-d]pyrimidin-3-yl]methyl]-4-fluorobenzonitrile | NA | 300000 | NA | NA | NA | NA | TTD |
| DPP9 | US11096924, DASH-inhibitors 5553 | NA | 2465000 | NA | NA | NA | NA | BindingDB |
| DPP9 | US11096924, DASH-inhibitors 5311 | NA | 5786000 | NA | NA | NA | NA | BindingDB |
| DPP9 | US11096924, DASH-inhibitors 5316 | NA | 468000 | NA | NA | NA | NA | BindingDB |
| DPP9 | US11096924, DASH-inhibitors 5323 | NA | 305000 | NA | NA | NA | NA | BindingDB |
| DPP9 | US11096924, DASH-inhibitors 5321 | NA | 112000 | NA | NA | NA | NA | BindingDB |
| DPP9 | US11096924, DASH-inhibitors 4160 | NA | 490000 | NA | NA | NA | NA | BindingDB |
| DPP9 | Glu-boroAla | NA | 7000000 | NA | NA | NA | NA | BindingDB |
| DPP9 | Sitagliptin | NA | 109100|130240 | NA | NA | NA | NA | BindingDB|PubChem |
| DPP9 | 1G244 | NA | 490000 | NA | NA | NA | NA | BindingDB |
| DPP9 | Talabostat | NA | 16000000 | NA | NA | NA | NA | BindingDB |
| DPP9 | Glu-boroSar | NA | 8400000 | NA | NA | NA | NA | BindingDB |
| DPP9 | (2S)-1-[(2S)-2-amino-3-(furan-3-yl)propanoyl]pyrrolidine-2-carbonitrile | NA | 288200 | NA | NA | NA | NA | TTD |
| DPP9 | (2S)-1-[(2S)-2-amino-3-pyridin-2-ylpropanoyl]pyrrolidine-2-carbonitrile | NA | 143600 | NA | NA | NA | NA | BindingDB|TTD |
| DRD1 | Imipenem | NA | NA | NA | NA | NA | 300000 | PubChem |
| DRD1 | Cefazolin | NA | NA | NA | NA | NA | 300000 | PubChem |
| DRD1 | Meropenem | NA | NA | NA | NA | NA | 300000 | PubChem |