| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| DPP7 |
2-Amino-1-(3-hydroxy-pyrrolidin-1-yl)-3-methyl-pentan-1-one |
NA |
299000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP7 |
2,6-Diamino-1-azetidin-1-yl-hexan-1-one |
NA |
159000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP7 |
Pyrrolidin-1-yl-(tetrahydro-thiophen-2-yl)-methanone |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| DPP7 |
2-Amino-1-(2,5-dihydro-pyrrol-1-yl)-3-methyl-pentan-1-one |
NA |
288000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP7 |
Benzoic acid 1-(2-amino-3-methyl-pentanoyl)-pyrrolidin-3-yl ester |
NA |
158000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP7 |
2-(Benzylamino)-1-cyclopentylethanethione |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| DPP7 |
benzyl (S)-5-amino-6-(1-(di-(4-acetamido)phenoxyphosphoryl)isoindolin-2-yl)-6- |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| DPP7 |
Anagliptin |
NA |
176700 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| DPP7 |
(2S,3R)-2-amino-3-hydroxy-1-(pyrrolidin-1-yl)butan-1-one |
NA |
230000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP7 |
(S)-2,6-diamino-1-(3,4-dihydroquinolin-1(2H)-yl)hexan-1-one |
NA |
393000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP7 |
(R)-(4-(1-amino-2-(2,4,5-trifluorophenyl)ethyl)piperidin-1-yl)(2,4-difluorophenyl)methanone |
NA |
11100000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP7 |
(R)-(4-(1-amino-2-(2,4,5-trifluorophenyl)ethyl)piperidin-1-yl)(isoquinolin-3-yl)methanone |
NA |
10200000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP7 |
(R)-(4-(1-amino-2-(2,4,5-trifluorophenyl)ethyl)piperidin-1-yl)(3-aminopyrazin-2-yl)methanone |
NA |
9110000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP7 |
2-Amino-3-methyl-1-(1-pyrrolidinyl)-1-butanone |
NA |
223000 |
NA |
NA |
NA |
NA |
BindingDB |
| DPP7 |
2-Amino-3-Methyl-1-Pyrrolidin-1-Yl-Butan-1-One |
NA |
153000|223000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| DPP7 |
Vaborbactam |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| DPP7 |
1G244 |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| DPP7 |
Vildagliptin |
NA |
1000000|500000 |
NA |
NA |
NA |
NA |
PubChem |
| DPP7 |
Talabostat |
NA|125000 |
10000000|NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| DPP7 |
(2S)-2-amino-N-(1-diphenoxyphosphorylethyl)-3-methyl-pentanamide |
NA |
116000 |
NA |
NA |
NA |
NA |
BindingDB |