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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
DPP7 (3S)-3-amino-4-(2-diphenoxyphosphorylpyrrolidin-1-yl)-4-oxo-butanamide NA 125000 NA NA NA NA TTD
DPP7 (2S)-2-amino-3-cyclohexyl-N-(1-diphenoxyphosphorylbutyl)propanamide NA 500000 NA NA NA NA BindingDB
DPP7 (2S)-2-amino-N-[cyclohexyl(diphenoxyphosphoryl)methyl]-3-(1H-imidazol-4-yl)propanamide NA 241000 NA NA NA NA BindingDB
DPP7 (3S)-3-amino-4-(2-diphenoxyphosphorylpyrrolidin-1-yl)-4-oxo-butanoic Acid NA 1000000 NA NA NA NA TTD
DPP7 cyclohexylglycine-(2S)-cyanopyrrolidine NA 102000 NA NA NA NA BindingDB
DPP7 (-)-(2S)-1-(((3-Hydroxytricyclo(3.3.1.1(3,7))dec-1-yl)amino)acetyl)pyrrolidine-2-carbonitrile NA 210000|500000 NA NA NA NA BindingDB|PubChem|TTD
DPP7 N-[diphenoxyphosphoryl(phenyl)methyl]-2-(isobutylamino)acetamide NA 158000 NA NA NA NA BindingDB
DPP7 1-[(1-Adamantylamino)acetyl]-2-pyrrolidinecarbonitrile NA 133500 NA NA NA NA BindingDB
DPP7 2-Oxo-2-pyrrolidin-1-ylethanamine NA 1000000 NA NA NA NA TTD
DPP7 (S)-3-amino-4-oxo-4-(pyrrolidin-1-yl)butanoic acid NA 500000 NA NA NA NA TTD
DPP7 (S)-3-amino-4-oxo-4-(pyrrolidin-1-yl)butanamide NA 152000 NA NA NA NA BindingDB|TTD
DPP7 N-Cyclohexyl-2-oxo-2-(1-pyrrolidinyl)ethaneamine NA 276000 NA NA NA NA BindingDB|TTD
DPP7 (1R)-2-[2-(1-adamantylamino)acetyl]cyclopentane-1-carbonitrile NA 133500 NA NA NA NA TTD
DPP7 N-Benzyl-2-oxo-2-(1-pyrrolidinyl)ethaneamine NA 500000 NA NA NA NA BindingDB|TTD
DPP7 (S)-2-amino-1-(pyrrolidin-1-yl)propan-1-one NA 179000 NA NA NA NA BindingDB|TTD
DPP7 (2S)-2-amino-1-(2-diphenoxyphosphorylpyrrolidin-1-yl)-3-hydroxy-propan-1-one NA 1000000 NA NA NA NA TTD
DPP7 Piperidine, 1-[[(phenylmethyl)amino]acetyl]- NA 397000 NA NA NA NA BindingDB|TTD
DPP7 (2S)-2-amino-1-(2-diphenoxyphosphorylpyrrolidin-1-yl)-3-methyl-butan-1-one NA 1000000 NA NA NA NA TTD
DPP7 (2S,4S)-1-[(3R)-3-amino-4-(2-chlorophenyl)butanoyl]-4-fluoropyrrolidine-2-carbonitrile NA 129710 NA NA NA NA BindingDB|TTD
DPP7 (2S,4S)-1-[(3R)-3-amino-4-(4-fluorophenyl)butanoyl]-4-fluoropyrrolidine-2-carbonitrile NA 192790 NA NA NA NA BindingDB|TTD