| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| EGFR |
(E)-3-[3-tert-butyl-4-hydroxy-5-[(2-methylpropan-2-yl)oxy]phenyl]-2-cyanoprop-2-enethioamide |
NA |
501187.23 |
NA |
NA |
NA |
NA |
TTD |
| EGFR |
5-naphthalen-1-ylsulfanyl-9H-pyrimido[4,5-b]indole-2,4-diamine |
NA |
167300 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| EGFR |
CID 138454747 |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| EGFR |
N-(2-hydroxyphenyl)-2-([1,3]thiazolo[3,2-a]benzimidazol-1-yl)acetamide |
NA |
55000000 |
NA |
NA |
NA |
NA |
BindingDB |
| EGFR |
4-N-[(4-chlorophenyl)methyl]-[1]benzofuro[2,3-b]pyridine-4,6-diamine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| EGFR |
4-N-[(4-methoxyphenyl)methyl]-[1]benzofuro[2,3-b]pyridine-4,6-diamine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| EGFR |
4-N-[(4-bromophenyl)methyl]-[1]benzofuro[2,3-b]pyridine-4,6-diamine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| EGFR |
N-[2-[[5-chloro-2-[[6-(3-hydroxyazetidin-1-yl)-2-methoxypyridin-3-yl]amino]pyrimidin-4-yl]amino]phenyl]methanesulfonamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| EGFR |
N-[2-[[5-chloro-2-[[6-(4-methylpiperazin-1-yl)-2-propan-2-yloxypyridin-3-yl]amino]pyrimidin-4-yl]amino]phenyl]methanesulfonamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| EGFR |
N-[2-[[5-chloro-2-[[6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methoxypyridin-3-yl]amino]pyrimidin-4-yl]amino]phenyl]methanesulfonamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| EGFR |
N-[2-[[5-chloro-2-[[2-methoxy-6-(4-methylpiperazin-1-yl)pyridin-3-yl]amino]pyrimidin-4-yl]amino]phenyl]cyclopropanesulfonamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| EGFR |
N-[2-[[5-chloro-2-[(2-methoxy-6-thiomorpholin-4-ylpyridin-3-yl)amino]pyrimidin-4-yl]amino]phenyl]methanesulfonamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| EGFR |
7,8-Dimethoxy-3-methyl-5,10-dihydro-3H-pyrimido[4,5-b]quinolin-4-one |
NA |
160000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| EGFR |
2-Cyano-3-(4-dimethylamino-phenyl)-acrylic acid |
NA|1400000 |
1400000|NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| EGFR |
2-Cyano-3-(4-fluorophenyl)acrylic acid |
833000|NA |
2500000|833000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| EGFR |
N-[4-methoxy-2-[methyl-[2-(methylamino)ethyl]amino]-5-[[4-(1-methylpyrrolo[3,2-b]pyridin-3-yl)pyrimidin-2-yl]amino]phenyl]prop-2-enamide |
NA |
277000 |
NA |
NA |
NA |
NA |
BindingDB |
| EGFR |
(2E)-2-Cyano-3-(4-methylphenyl)prop-2-enoic acid |
NA|1350000 |
1350000|NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| EGFR |
Azd-1152hqpa |
NA |
NA |
980000 |
NA |
NA |
NA |
BindingDB |
| EGFR |
Egfr-IN-51 |
NA |
102600|461630 |
NA |
NA |
NA |
NA |
BindingDB |
| EGFR |
N-(5-tert-butyl-2-methylpyrazol-3-yl)-2-[4-[[6-(1-methylpyrazol-4-yl)thieno[3,2-d]pyrimidin-4-yl]amino]phenyl]acetamide |
NA |
176090 |
NA |
NA |
NA |
NA |
BindingDB |