| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| EGFR |
2-[(5-fluoro-2-hydroxyphenyl)-(3-oxo-1H-isoindol-2-yl)methyl]-3H-quinazolin-4-one |
NA |
5300000 |
NA |
NA |
NA |
NA |
BindingDB |
| EGFR |
(E)-N-[2-[2-(dimethylamino)ethyl-methylamino]-4-methoxy-5-[[4-methyl-5-(1-methylindol-2-yl)pyrimidin-2-yl]amino]phenyl]hex-2-enamide |
NA |
191300 |
NA |
NA |
NA |
NA |
BindingDB |
| EGFR |
SB 203580 |
NA |
NA |
1900000 |
NA |
NA |
NA |
BindingDB |
| EGFR |
Erlotinib |
NA |
421000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| EGFR |
N-[5,21-dihydroxy-12,14-dioxo-3-[3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]-3,13,23-triazahexacyclo[14.7.0.02,10.04,9.011,15.017,22]tricosa-1,4(9),5,7,10,15,17(22),18,20-nonaen-13-yl]formamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| EGFR |
Piperonylidenemalononitrile |
117000 |
350000|NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| EGFR |
Malononitrile, furfurylidene- |
NA |
1250000 |
NA |
NA |
NA |
NA |
TTD |
| EGFR |
13-Amino-5,21-dihydroxy-3-[3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]-3,13,23-triazahexacyclo[14.7.0.02,10.04,9.011,15.017,22]tricosa-1,4(9),5,7,10,15,17(22),18,20-nonaene-12,14-dione |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| EGFR |
AG 126 |
150000 |
450000|NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| EGFR |
Tyrphostin A1 |
400000 |
NA |
NA |
NA |
NA |
NA |
GtoPDB|TTD |
| EGFR |
Lapatinib |
NA |
377400 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| EGFR |
1-(1,3-Benzodioxol-5-yl)-3-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)thiourea |
NA |
432670 |
NA |
NA |
NA |
NA |
BindingDB |
| EGFR |
2-(4-Methoxybenzoyl)propanedinitrile |
NA |
450000 |
NA |
NA |
NA |
NA |
BindingDB |
| EGFR |
[(e)-(4-Methoxyphenyl)diazenyl]propanedinitrile |
NA |
600000 |
NA |
NA |
NA |
NA |
BindingDB |
| EGFR |
Malononitrile, (3-pyridylmethylene)- |
NA |
225000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| EGFR |
N-[(2R,3S,4S,6S)-3-methoxy-2-methyl-16-oxo-29-oxa-1,7,17-triazaoctacyclo[12.12.2.12,6.07,28.08,13.015,19.020,27.021,26]nonacosa-8,10,12,14,19,21,23,25,27-nonaen-4-yl]-N-methylbenzamide |
NA |
NA |
760000 |
NA |
NA |
NA |
BindingDB |
| EGFR |
2-(2-Oxoindolin-3-ylidene)malononitrile |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| EGFR |
Metachromin L |
NA |
490000 |
NA |
NA |
NA |
NA |
BindingDB |
| EGFR |
N4-(4-fluoro-3-(trifluoromethyl)phenyl)-6-phenethyl-7H-pyrrolo[2,3-d]pyrimidine-2,4-diamine |
NA |
122000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| EGFR |
6-phenethyl-N4-(3-(trifluoromethyl)phenyl)-7H-pyrrolo[2,3-d]pyrimidine-2,4-diamine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |