| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| EGFR |
2-[(3-Hydroxyphenyl)methylidene]propanedinitrile |
123000 |
375000|NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| EGFR |
2-(1H-pyrrol-2-ylmethylene)malononitrile |
NA |
260000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| EGFR |
(3,5-Dimethoxybenzylidene)propanedinitrile |
400000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| EGFR |
Tandutinib |
NA |
NA |
400000 |
NA |
NA |
NA |
BindingDB |
| EGFR |
Dasatinib |
NA |
NA |
120000 |
NA |
NA |
NA |
BindingDB |
| EGFR |
(4-Morpholin-4-ylbenzylidene)malononitrile |
250000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| EGFR |
Cefazolin |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| EGFR |
N-(4-(2,2-Dicyanovinyl)phenyl)acetamide |
NA |
325000 |
NA |
NA |
NA |
NA |
TTD |
| EGFR |
2-(4-Fluorobenzylidene)malononitrile |
400000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| EGFR |
MALONONITRILE, (p-CYANOBENZYLIDENE)- |
NA |
1400000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| EGFR |
2-((3,5-di-tert-Butyl-4-hydroxyphenyl)-methylene)-4-cyclopentene-1,3-dione |
NA |
320000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| EGFR |
Meropenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| EGFR |
2,4-Diaminofuro[2,3-d]pyrimidine, 2 |
NA |
160300 |
NA |
NA |
NA |
NA |
BindingDB |
| EGFR |
5-[(1z)-2-(2-Methoxyphenyl)-3-Methylbut-1-En-1-Yl]furo[2,3-D]pyrimidine-2,4-Diamine |
NA |
111400 |
NA |
NA |
NA |
NA |
BindingDB |
| EGFR |
2,4-Diaminofuro[2,3-d]pyrimidine, 5 |
NA |
529300 |
NA |
NA |
NA |
NA |
BindingDB |
| EGFR |
2,4-Diaminofuro[2,3-d]pyrimidine, 12 |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| EGFR |
2,4-Diaminofuro[2,3-d]pyrimidine, 13 |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| EGFR |
Staurosporine |
NA |
178000 |
NA |
NA |
NA |
NA |
BindingDB |
| EGFR |
13-(Ethylamino)-5,21-dihydroxy-3-[3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]-3,13,23-triazahexacyclo[14.7.0.02,10.04,9.011,15.017,22]tricosa-1,4(9),5,7,10,15,17(22),18,20-nonaene-12,14-dione |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| EGFR |
13-(Dimethylamino)-5,21-dihydroxy-3-[3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]-3,13,23-triazahexacyclo[14.7.0.02,10.04,9.011,15.017,22]tricosa-1,4(9),5,7,10,15,17(22),18,20-nonaene-12,14-dione |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |