| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ELANE |
4-Hydroxy-6-undecyl-1H-pyridin-2-one |
NA |
153000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ELANE |
2-Butyl-2-(3,5-dibutyl-4-hydroxy-6-oxopyran-2-yl)octanal |
151356|151356.12 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ELANE |
4-Hydroxy-3-methyl-6-phenacylpyran-2-one |
977237|977237.22 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ELANE |
3,5-dibutyl-4-hydroxy-6-[(E)-1-phenylprop-1-enyl]pyran-2-one |
363078|363078.05 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ELANE |
4-Hydroxy-6-nonyl-pyran-2-one |
400000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ELANE |
Vaborbactam |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| ELANE |
(2S)-2-[[(2R)-2-[[(2S)-6-(adamantane-1-carbonylamino)-2-[[(2S,3R)-2-(benzylamino)-3-methylpentanoyl]amino]hexanoyl]amino]-3-sulfanylpropanoyl]amino]-3-methylbutanoic acid |
269700 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ELANE |
|
207000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ELANE |
|
199000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ELANE |
|
113000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ELANE |
(4R)-4-[[(2S)-2-acetamido-3-carboxypropanoyl]amino]-5-[[(2S,3S)-3-methyl-1-[[(2S)-3-methyl-1-[(2S,4R)-2-[[methyl-[[(1S)-1-phenylethyl]carbamoyl]amino]carbamoyl]-4-phenylmethoxypyrrolidin-1-yl]-1-oxobutan-2-yl]amino]-1-oxopentan-2-yl]amino]-5-oxopentanoic acid |
NA |
168000 |
NA |
NA |
NA |
NA |
TTD |
| ELANE |
(4R)-4-[[(2S)-2-acetamido-3-carboxypropanoyl]amino]-5-[[(2S,3S)-3-methyl-1-[[(2S)-3-methyl-1-oxo-1-[(2S,4R)-2-[[pentyl-[[(1S)-1-phenylethyl]carbamoyl]amino]carbamoyl]-4-phenylmethoxypyrrolidin-1-yl]butan-2-yl]amino]-1-oxopentan-2-yl]amino]-5-oxopentanoic acid |
NA |
151000 |
NA |
NA |
NA |
NA |
TTD |
| ELANE |
5-Methyl-3-(4-nitrophenyl)-1,3-oxazolidine-2,4-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| ELANE |
3-(4-Methoxyphenyl)-5,5-dimethyl-1,3-oxazolidine-2,4-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| ELANE |
5,5-Dimethyl-3-(4-nitrophenyl)-1,3-oxazolidine-2,4-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| ELANE |
3-(4-Methoxyphenyl)-5-methyl-1,3-oxazolidine-2,4-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| ELANE |
Ac-Ile-Leu-Gly-NHBu |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ELANE |
Tfa-Ile-Leu-Gly-NHBu |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ELANE |
(2S,3S)-2-acetamido-N-[(1R)-1-[[3-(butylamino)-3-oxopropyl]-dihydroxysilyl]-3-methylbutyl]-3-methylpentanamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ELANE |
N-[3-[(2-fluorophenyl)methoxy]phenyl]-1-pyridin-4-ylpiperidine-4-carboxamide |
250000 |
NA |
NA |
NA |
NA |
NA |
TTD |