| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ELANE |
N-[3-[(3,5-difluorophenyl)methoxy]phenyl]-1-pyridin-4-ylpiperidine-4-carboxamide |
250000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| ELANE |
N-[3-[(3,4-dimethoxyphenyl)methoxy]phenyl]-1-pyridin-4-ylpiperidine-4-carboxamide |
250000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| ELANE |
(3S)-3-acetamido-4-[[(2R)-1-[[(2S,3S)-1-[[(2S)-1-[(2S)-2-[[(3S)-1-(benzylamino)-1,2-dioxohexan-3-yl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]amino]-3-methyl-1-oxopentan-2-yl]amino]-3-carboxy-1-oxopropan-2-yl]amino]-4-oxobutanoic acid |
NA |
172000 |
NA |
NA |
NA |
NA |
BindingDB |
| ELANE |
(R)-3-((S)-2-Acetylamino-3-carboxy-propionylamino)-N-((1S,2S)-1-{(S)-1-[2-((R)-1-benzylcarbamoyl-butylcarbamoyl)-pyrrolidine-1-carbonyl]-2-methyl-propylcarbamoyl}-2-methyl-butyl)-succinamic acid |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ELANE |
(R)-2-{[1-((S)-2-{(2S,3S)-2-[(R)-2-((S)-2-Acetylamino-3-carboxy-propionylamino)-3-carboxy-propionylamino]-3-methyl-pentanoylamino}-3-methyl-butyryl)-pyrrolidine-2-carbonyl]-amino}-pentanoic acid benzyl ester |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ELANE |
2-(4-(2,5-dimethyl-1H-pyrrol-1-yl)phenyl)acetic acid |
NA |
124900 |
NA |
NA |
NA |
NA |
TTD |
| ELANE |
2-chloro-5-(2,5-dimethyl-1H-pyrrol-1-yl)benzoic acid |
NA |
160200 |
NA |
NA |
NA |
NA |
TTD |
| ELANE |
[4-[[2-[(E)-N-hydroxy-C-methylcarbonimidoyl]phenyl]sulfamoyl]phenyl] 2,2-dimethylpropanoate |
NA |
221560 |
NA |
NA |
NA |
NA |
BindingDB |
| ELANE |
2-Hydroxy-3-(4-methoxy-6-oxo-6H-pyran-2-yl)-acrylic acid pentyl ester |
410000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ELANE |
(S)-N1-(2-Benzylcarbamoyl-1-methyl-2-oxoethyl)-2-[(S)-2-(3,3-dimethyl-butanoylamino)-3,3-dimethyl-butanoylamino]-N4,N4-dimethylsuccinamide |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| ENGASE |
(2S,3S)-3-Hydroxybaikiain |
NA |
750000 |
NA |
NA |
NA |
NA |
BindingDB |
| ENPP1 |
|
NA|850000 |
900000|NA |
NA |
NA |
NA |
NA |
BindingDB |
| ENPP1 |
5-bromo-N-naphthalen-2-ylsulfonylpyrrolo[2,3-b]pyridine-1-carboxamide |
NA |
177500 |
NA |
NA |
NA |
NA |
BindingDB |
| ENPP1 |
(4-(((6,7-Dimethoxyquinazolin-4-yl)oxy)methyl)phenyl)(imino)(methyl)-lambda6-sulfanone |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB |
| ENPP1 |
Imino(4-((8-methoxyquinazolin-4-yl)oxy)phenyl)(methyl)-lambda6-sulfanone |
NA|210000 |
1300000|NA |
NA |
NA |
NA |
NA |
BindingDB |
| ENPP1 |
(4-(Cinnolin-4-yloxy)phenyl)(imino)(methyl)-lambda6-sulfanone |
NA|310000 |
1200000|NA |
NA |
NA |
NA |
NA |
BindingDB |
| ENPP1 |
6-methyl-4-(4-(S-methylsulfonimidoyl)phenoxy)quinoline-3-carbonitrile |
NA |
2600000 |
NA |
NA |
NA |
NA |
BindingDB |
| ENPP1 |
(2-(1-(7,8-Dimethoxyquinazolin-4-yl)piperidin-4-yl)ethyl)(imino)(methyl)-l6-sulfanone |
1400000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| ENPP1 |
Imino(4-{[(8-methoxyquinolin-4-yl)oxy]methyl}phenyl)methyl-lambda6-sulfanone |
NA |
1100000 |
NA |
NA |
NA |
NA |
BindingDB |
| ENPP1 |
(3-Bromo-4-{[(7-methoxyquinolin-4-yl)oxy]methyl}phenyl)(imino)methyl-lambda6-sulfanone |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |