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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ENPP1 Imino(4-(7-methoxyquinolin-4-yl)benzyl)(methyl)-lambda6-sulfanone NA 920000 NA NA NA NA BindingDB
ENPP1 Imino(2-(1-(8-methoxyquinazolin-4-yl)piperidin-4-yl)ethyl)(methyl)-lambda6-sulfanone NA|180000 120000|880000|NA NA NA NA NA BindingDB
ENPP1 1-(1-Imino-1-oxido-1lambda6-thiomorpholino)-2-(7-methoxyquinolin-4-yl)ethan-1-one NA 8800000 NA NA NA NA BindingDB
ENPP1 Imino({4-[(8-methoxyquinolin-4-yl)oxy]phenyl})methyl-lambda6-sulfanone NA 160000 NA NA NA NA BindingDB
ENPP1 Imino(methyl){2-[1-(quinolin-4-yl)piperidin-4-yl]ethyl}-lambda6-sulfanone NA|410000 1400000|NA NA NA NA NA BindingDB
ENPP1 {[1-(3-Fluoro-8-methoxyquinolin-4-yl)piperidin-4-yl]methyl}(imino)methyl-lambda6-sulfanone 370000 NA NA NA NA NA BindingDB
ENPP1 Imino(4-(7-methoxyquinolin-4-yl)phenethyl)(methyl)-lambda6-sulfanone NA 140000 NA NA NA NA BindingDB
ENPP1 Imino({4-[(6-methoxy-1,5-naphthyridin-4-yl)oxy]phenyl})methyl-lambda6-sulfanone NA 8100000 NA NA NA NA BindingDB
ENPP1 Imino[7-(8-methoxyquinazolin-4-yl)-1,7-diazaspiro[3.5]nonan-1-yl]methyl-lambda6-sulfanone 110000 NA NA NA NA NA BindingDB
ENPP1 Imino({2-[4-(8-methoxyquinazolin-4-yl)phenyl]ethyl})methyl-lambda6-sulfanone NA 1800000 NA NA NA NA BindingDB
ENPP1 {4-[(6,7-Dimethoxyquinolin-4-yl)oxy]-3-fluorophenyl}(imino)methyl-lambda6-sulfanone NA 220000 NA NA NA NA BindingDB
ENPP1 {4-[(8-Fluoro-7-methoxyquinolin-4-yl)oxy]phenyl}(imino)methyl-lambda6-sulfanone NA 310000 NA NA NA NA BindingDB
ENPP1 Imino(methyl)[4-(quinolin-4-yloxy)phenyl]-lambda6-sulfanone NA|110000 340000|NA NA NA NA NA BindingDB
ENPP1 {5-[(6,7-Dimethoxyquinolin-4-yl)oxy]pyridin-2-yl}(imino)methyl-lambda6-sulfanone NA 260000 NA NA NA NA BindingDB
ENPP1 Imino({3-[(7-methoxyquinolin-4-yl)oxy]phenyl})methyl-lambda6-sulfanone NA 180000 NA NA NA NA BindingDB
ENPP1 Imino-[4-(7-methoxyquinolin-4-yl)oxyphenyl]-methyl-oxo-lambda6-sulfane NA 180000 NA NA NA NA BindingDB
ENPP1 Cyclopropyl-imino-[4-(7-methoxyquinolin-4-yl)oxyphenyl]-oxo-lambda6-sulfane NA 520000 NA NA NA NA BindingDB
ENPP1 imino-[7-(7-methoxyquinolin-4-yl)-3,4-dihydro-1H-isoquinolin-2-yl]-methyl-oxo-lambda6-sulfane 110000 NA NA NA NA NA BindingDB
ENPP1 Imino(4-((7-methoxy-1,5-naphthyridin-4-yl)oxy)phenyl)(methyl)-lambda6-sulfanone NA 23000000 NA NA NA NA BindingDB
ENPP1 (4-((6,7-Dimethoxyquinazolin-4-yl)oxy)phenyl)(imino)(methyl)-lambda6-sulfanone NA 180000 NA NA NA NA BindingDB