| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| F10 |
3-Carbamimidoylbenzamide |
250000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
naphth-2-ylsulfonyl-Phe(3-amidino)-Pro-OH |
130000|130016.96 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
2-amino-5-[(3-hydroxynaphthalene-2-)amido]-1H-1,3-benzodiazol-3-ium |
200000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| F10 |
3-(Benzyl(2-(4-carbamimidoylbenzyl)-4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)amino)-3-oxopropanoic acid |
139000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
3-[2-(4-Carbamimidoylbenzyloxy)-4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazine-7-carbonylamino]propanoic acid |
112000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
Ethyl 2-(benzyl{2-[(4-carbamimidoylphenoxy)methyl]-2,4-dimethyl-3,4-dihydro-2H-1,4-benzoxazin-7-yl}amino)-2-oxoacetate |
112000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
N-{3-[(4-fluorobenzyl)oxy]-phenyl}piperidine-3-carboxamide |
260000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
N-(4-(biphenyl-4-ylmethoxy)phenyl)piperidine-4-carboxamide |
126000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
4-(Aminomethyl)benzenecarboximidamide |
680000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL|TTD |
| F10 |
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-(2-methylindol-1-yl)acetate |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| F10 |
N-(4-Carbamimidoyl-3-choro-phenyl)-2-hydroxy-3-iodo-5-methyl-benzamide |
110000|115000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
2-Chloro-benzenesulfonic acid 3-(5-guanidino-pentyloxy)-5-methyl-phenyl ester |
120000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
2-Chloro-benzenesulfonic acid 3-(3-guanidino-propoxy)-5-methyl-phenyl ester |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F10 |
2-Chloro-benzenesulfonic acid 3-(4-guanidino-butoxy)-5-methyl-phenyl ester |
110000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
methyl 2-[(1R,3aS,8bS)-1-(5-amino-5-iminopentyl)-2-oxo-1,3a,4,8b-tetrahydroindeno[2,1-b]pyrrol-3-yl]acetate |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| F10 |
5-[(1R,3aS,8bS)-2-oxo-3,3a,4,8b-tetrahydro-1H-indeno[2,1-b]pyrrol-1-yl]pentanimidamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| F10 |
3-[3-(3-Benzyl-1H-indol-2-yl)-5-bromo-4-hydroxy-phenyl]-propionic acid |
300000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
5-Bromo-N-(4-guanidino-phenyl)-2-hydroxy-benzamide |
470000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F10 |
N-(4-Guanidino-phenyl)-2-hydroxy-5-nitro-benzamide |
470000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F10 |
N-(4-Guanidino-phenyl)-2-hydroxy-benzamide |
104000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |