| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| F10 |
N-(2-Amino-4,5,6,7-tetrahydro-benzothiazol-6-yl)-2-[6-methyl-2-oxo-3-(propane-1-sulfonylamino)-2H-pyridin-1-yl]-acetamide |
200000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
N-(2-Amino-4,5,6,7-tetrahydro-benzothiazol-6-yl)-2-[3-(butane-1-sulfonylamino)-6-methyl-2-oxo-2H-pyridin-1-yl]-acetamide |
179000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
2-(6-Methyl-2-oxo-3-p-tolylmethanesulfonylamino-2H-pyridin-1-yl)-N-(4,5,6,7-tetrahydro-2H-indazol-5-ylmethyl)-acetamide |
228000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
N-((R)-2-Amino-4,5,6,7-tetrahydro-benzothiazol-6-yl)-2-[3-(4-fluoro-phenylmethanesulfonylamino)-6-methyl-2-oxo-2H-pyridin-1-yl]-acetamide |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F10 |
N-(3-Amino-2-imino-2,3,4,5,6,7-hexahydro-benzothiazol-6-yl)-2-(6-methyl-2-oxo-3-phenylmethanesulfonylamino-2H-pyridin-1-yl)-acetamide |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F10 |
N-((S)-2-Amino-4,5,6,7-tetrahydro-benzothiazol-6-yl)-2-[3-(4-fluoro-phenylmethanesulfonylamino)-6-methyl-2-oxo-2H-pyridin-1-yl]-acetamide |
176400 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
N-(3-Amino-2-imino-2,3,4,5,6,7-hexahydro-benzothiazol-6-yl)-2-[3-(4-fluoro-phenylmethanesulfonylamino)-6-methyl-2-oxo-2H-pyridin-1-yl]-acetamide |
131000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
N-((S)-2-Amino-4,5,6,7-tetrahydro-benzothiazol-6-yl)-2-(6-methyl-2-oxo-3-phenylmethanesulfonylamino-2H-pyridin-1-yl)-acetamide |
370600 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
2-[6-Methyl-2-oxo-3-(3-trifluoromethyl-phenylmethanesulfonylamino)-2H-pyridin-1-yl]-N-(4,5,6,7-tetrahydro-2H-indazol-5-ylmethyl)-acetamide |
252000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
(2S)-1-[(2R)-2-amino-3,3-diphenylpropanoyl]-N-[1-(diaminomethylideneamino)-5,8-dioxo-8-piperidin-1-yloctan-4-yl]pyrrolidine-2-carboxamide |
149000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
(S)-1-(3-Phenyl-3-pyridin-4-yl-propionyl)-pyrrolidine-2-carboxylic acid (4-amino-cyclohexylmethyl)-amide; TFA |
400000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
(S)-1-(3-Phenyl-3-pyridin-3-yl-propionyl)-pyrrolidine-2-carboxylic acid (4-amino-cyclohexylmethyl)-amide; TFA |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F10 |
(S)-1-(3-Phenyl-3-pyridin-2-yl-propionyl)-pyrrolidine-2-carboxylic acid (4-amino-cyclohexylmethyl)-amide; TFA |
370000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
(S)-1-(3-Benzo[1,3]dioxol-5-yl-3-pyridin-3-yl-propionyl)-pyrrolidine-2-carboxylic acid (4-amino-cyclohexylmethyl)-amide; TFA |
1000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
3-[(2S)-2-[(4-methoxy-2,3,6-trimethylphenyl)sulfonylamino]-3-(4-methylsulfonylpiperazin-1-yl)-3-oxopropyl]benzenecarboximidamide |
119000|119949.93 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
quinolin-8-ylsufonyl-Phe(3-amidino)-piperidino(4-Me) |
179000|179887.09 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
(2S)-3-(3-carbamimidoylphenyl)-2-(naphthalen-2-ylsulfonylamino)-N-propan-2-ylpropanamide |
359000|359749.34 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
(3S)-4-(3-carbamimidoylphenyl)-3-(naphthalen-2-ylsulfonylamino)-2-oxobutanoic acid |
130000|130016.96 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
3-[(2S)-2-amino-3-(4-methylpiperidin-1-yl)-3-oxopropyl]benzenecarboximidamide |
230000|230144.18 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
naphth-2-ylsulfonyl-Phe(3-amidino)-Pro-OMe |
109000|109900.58 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |