| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| F10 |
Methyl-phe-pro-amino-cyclohexylglycine |
1000000 |
NA |
NA |
NA |
NA |
NA |
PubChem|TTD |
| F10 |
(S)-N-((1-carbamimidoylpiperidin-4-yl)methyl)-5-guanidino-2-((S)-2-((S)-5-guanidino-2-(2-phenylacetamido)pentanamido)-3-methylbutanamido)pentanamide |
123000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
(2R)-2-amino-N-[3,5-bis[(E)-N-(diaminomethylideneamino)-C-methylcarbonimidoyl]phenyl]-5-(diaminomethylideneamino)pentanamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
N-(3,5-bis(-1-(2-carbamimidoylhydrazono)ethyl)phenyl)-5-guanidinopentanamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
N-(3,5-bis(-1-(2-carbamimidoylhydrazono)ethyl)phenyl)-6-guanidinohexanamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
amino-N-(3,5-bis(-1-(2-carbamimidoylhydrazono)ethyl)phenyl)butanamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
Mangiferin heptasulfate |
NA |
970000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
Sodium;[3-ethoxycarbonyl-2-[(3-ethoxycarbonyl-6-methoxy-2-methyl-1-benzofuran-5-yl)oxymethyl]-6-methoxy-1-benzofuran-5-yl] sulfate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| F10 |
Boc-Darg-Gly-Arg-Cho |
NA |
180000 |
NA |
NA |
NA |
NA |
BindingDB |
| F10 |
Thieno(2,3-B)Pyridine-2-Carboxamidine |
360000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| F10 |
Ac-Tyr-Thr-hArg-Bn |
NA |
1078000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
BnSO2-Phe-Leu-hArg-Bn |
NA |
580000 |
NA |
NA |
NA |
NA |
TTD |
| F10 |
H-Phe-Phe-hArg-Bn |
NA |
1480000 |
NA |
NA |
NA |
NA |
TTD |
| F10 |
BnSO2-Phe-Phe-hArg-Bn |
NA |
590000 |
NA |
NA |
NA |
NA |
TTD |
| F10 |
H-Tyr-Thr-hArg-Bn |
NA |
1340000 |
NA |
NA |
NA |
NA |
TTD |
| F10 |
Ac-Phe-Phe-hArg-Bn |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| F10 |
Cbz-D-Phe-Phe-hArg-Bn |
NA |
440000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
BnSO2-D-Phe-Phe-hArg-Bn |
NA |
640000 |
NA |
NA |
NA |
NA |
TTD |
| F10 |
Cbz-Phe-Phe-hArg-Bn |
NA |
508000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
6-amino-N-[(3S,7E,9S,12R,16S,19S)-16-[[3-(aminomethyl)phenyl]methyl]-12-[(2S)-butan-2-yl]-9-[(4-hydroxyphenyl)methyl]-2,6,11,14,18-pentaoxo-1,5,10,13,17-pentazabicyclo[17.3.0]docos-7-en-3-yl]hexanamide |
360000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |