| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| F10 |
ethyl 1-[4-[(5R)-5-[[(2-amino-1,3-thiazole-5-carbonyl)amino]methyl]-2-oxo-1,3-oxazolidin-3-yl]phenyl]piperidine-4-carboxylate |
111000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
N-[3-[(4-fluorophenyl)methoxy]phenyl]-1-propan-2-ylpiperidine-4-carboxamide |
250000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F10 |
N-[2-[(3-fluorophenyl)methoxy]phenyl]-1-pyridin-4-ylpiperidine-4-carboxamide |
250000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F10 |
N-[3-[(3-chlorophenyl)methoxy]phenyl]-1-pyridin-4-ylpiperidine-4-carboxamide |
250000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F10 |
N-[3-[(3,5-dimethoxyphenyl)methoxy]phenyl]-1-pyridin-4-ylpiperidine-4-carboxamide |
126000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
N-[3-[(3-fluorophenoxy)methyl]phenyl]-1-pyridin-4-ylpiperidine-4-carboxamide |
250000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F10 |
4-Amino-4-{[(4-carbamimidoyl-benzylcarbamoyl)-methyl]-carbamoyl}-butyric acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F10 |
(2R)-2-(benzylcarbamoylamino)-5-(diaminomethylideneamino)-N-[2-[[(2S)-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-2-oxoethyl]pentanamide |
NA |
170000 |
NA |
NA |
NA |
NA |
BindingDB |
| F10 |
[2-[(3,5-Dimethyl-1-phenylpyrazol-4-yl)amino]-2-oxoethyl] 2-(4-methyl-2-oxo-1,3-thiazol-3-yl)acetate |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| F10 |
Argatroban |
NA |
134000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| F10 |
2-(6-Methyl-2-oxo-3-phenylmethanesulfonylamino-2H-pyridin-1-yl)-N-(4,5,6,7-tetrahydro-2H-indazol-5-ylmethyl)-acetamide |
103000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
2-(2,6-Difluorophenyl)pyrido[3,4-d][1,3]oxazin-4-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| F10 |
1-Methyl-6-(2-methylphenyl)pyrazolo[3,4-d][1,3]oxazin-4-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| F10 |
7-Ethylsulfanyl-2-(2-fluorophenyl)pyrimido[4,5-d][1,3]oxazin-4-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| F10 |
2-(2,6-Difluorophenyl)-7-(trifluoromethyl)-4H-3,1-benzoxazine-4-one |
NA |
174000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F10 |
(2S)-2-amino-N-[2-[(4-carbamimidoylphenyl)methylamino]-2-oxoethyl]-3-hydroxypropanamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F10 |
2-Amino-N-[(4-carbamimidoyl-benzylcarbamoyl)-methyl]-3-hydroxy-propionamide |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F11 |
H-Cys(1)-Pro-Ala-Tyr-Ser-Arg-Tyr-Leu-Asp-Cys(1)-OH |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F11 |
Sodium;[2-[[6-methoxy-3-[(2-methylpropan-2-yl)oxycarbonyl]-1-benzofuran-5-yl]oxymethyl]-1,3-benzothiazol-6-yl] sulfate |
NA |
124000 |
NA |
NA |
NA |
NA |
TTD |
| F11 |
sodium;[2-[(2-benzyl-3-ethoxycarbonyl-6-methoxy-1-benzofuran-5-yl)oxymethyl]-3-ethoxycarbonyl-1H-indol-5-yl] sulfate |
NA |
118000 |
NA |
NA |
NA |
NA |
TTD |