| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| F11 |
N-[(S)-4-guanidino-1-(thiazole-2-carbonyl)-butyl]-3-methyl-butyramide |
NA |
123000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F11 |
naphthalene-2-carboxylic acid [(S)-4-guanidino-1-(thiazole-2-carbonyl)-butyl]-amide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| F11 |
naphthalene-1-sulfonic acid [(S)-4-guanidino-1-(thiazole-2-carbonyl)-butyl]-amide |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F11 |
N-[(S)-4-guanidino-1-(thiazole-2-carbonyl)-butyl]-2-naphthalen-1-yl-acetamide |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| F11 |
N-[(2S)-6-amino-1-[5-[[4-[2-(3,4-dichlorophenyl)ethoxy]phenyl]methyl]-1,2,4-oxadiazol-3-yl]-1-oxohexan-2-yl]-3,4-difluorobenzamide |
150000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F11 |
(1R,6S,8S,8aS)-6-amino-N-[(4-carbamimidoylphenyl)methyl]-1-ethyl-8-methoxy-6-(2-methylprop-2-enyl)-5-oxo-1,2,3,7,8,8a-hexahydroindolizine-3-carboxamide;(E)-but-2-enedioic acid |
NA |
133000 |
NA |
NA |
NA |
NA |
TTD |
| F11 |
N-((R)-2-((S)-1-((2-allyl-5-chloro-1H-indol-3-yl)methylamino)-4-methyl-1-oxopentan-2-ylamino)-1-cyclohexyl-2-oxoethyl)pent-4-enamide |
NA |
103100 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F11 |
(3E,9R,12S)-19-chloro-9-cyclohexyl-12-(2-methylpropyl)-7,7-dioxo-7lambda6-thia-8,11,14,23-tetrazatricyclo[14.7.0.017,22]tricosa-1(16),3,17(22),18,20-pentaene-10,13-dione |
NA |
767800 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F11 |
(S)-N-((R)-2-((S)-1-((2-allyl-5-chloro-1H-indol-3-yl)methylamino)-4-methyl-1-oxopentan-2-ylamino)-1-cyclohexyl-2-oxoethyl)-2-phenylpent-4-enamide |
NA |
145900 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F11 |
(9R,12S)-19-chloro-9-cyclohexyl-12-(2-methylpropyl)-7,7-dioxo-7lambda6-thia-8,11,14,23-tetrazatricyclo[14.7.0.017,22]tricosa-1(16),17(22),18,20-tetraene-10,13-dione |
NA |
175900 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F11 |
(3E,6S,9R,12S)-19-chloro-9-cyclohexyl-12-(2-methylpropyl)-6-phenyl-8,11,14,23-tetrazatricyclo[14.7.0.017,22]tricosa-1(16),3,17(22),18,20-pentaene-7,10,13-trione |
NA |
135800 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F11 |
N-[(6-Amino-2,4-Dimethylpyridin-3-Yl)methyl]-1-({4-[(1h-Pyrazol-1-Yl)methyl]phenyl}methyl)-1h-Pyrazole-4-Carboxamide |
NA |
106000 |
NA |
NA |
NA |
NA |
BindingDB |
| F11 |
(3R)-2-[2-(4-chlorophenyl)acetyl]-N-[4-(3-oxomorpholin-4-yl)phenyl]-3,4-dihydro-1H-isoquinoline-3-carboxamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| F11 |
2-(3-Cyano-4-methoxyphenyl)-3-hydroxy-5-methylimidazole-4-carboxylic acid |
243000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| F11 |
[4-(5-Methoxy-4-oxo-3,7-disulfooxychromen-2-yl)-2-[[1-[4-[4-oxo-2-(3-sulfooxyphenyl)quinazolin-3-yl]butyl]triazol-4-yl]methoxy]phenyl] hydrogen sulfate |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| F11 |
[2-Methoxy-4-[3-[4-[4-[[5-(5-methoxy-4-oxo-3,7-disulfooxychromen-2-yl)-2-sulfooxyphenoxy]methyl]triazol-1-yl]butyl]-4-oxoquinazolin-2-yl]phenyl] hydrogen sulfate |
NA |
216000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F11 |
[3-[3-[4-[4-[[5-(5-Methoxy-4-oxo-3,7-disulfooxychromen-2-yl)-2-sulfooxyphenoxy]methyl]triazol-1-yl]butyl]-4-oxoquinazolin-2-yl]-5-sulfooxyphenyl] acetate |
NA |
407000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F11 |
[4-[4-Oxo-3-[[1-[2-[4-[[4-oxo-2-(4-sulfooxyphenyl)quinazolin-3-yl]methyl]triazol-1-yl]ethyl]triazol-4-yl]methyl]quinazolin-2-yl]phenyl] hydrogen sulfate |
NA |
305000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| F11 |
[3-[4-Oxo-3-[[1-[4-[4-oxo-2-(3-sulfooxyphenyl)quinazolin-3-yl]butyl]triazol-4-yl]methyl]quinazolin-2-yl]phenyl] acetate |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| F11 |
[3-[4-Oxo-3-[[1-[4-[4-oxo-2-(3-sulfooxyphenyl)quinazolin-3-yl]butyl]triazol-4-yl]methyl]quinazolin-2-yl]phenyl] hydrogen sulfate |
NA |
102000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |