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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
F13A1 (2S)-5-oxo-2-[[(2S)-3-phenyl-2-(phenylmethoxycarbonylamino)propanoyl]amino]-6-(1,4,5-trimethyl-3-phenylimidazol-1-ium-2-yl)sulfanylhexanoic acid;bromide NA 200000 NA NA NA NA TTD
F13A1 (2S)-5-oxo-2-[[2-(phenylmethoxycarbonylamino)acetyl]amino]-6-(1,4,5-trimethyl-3-phenylimidazol-1-ium-2-yl)sulfanylhexanoic acid;bromide NA 200000 NA NA NA NA TTD
F13A1 (2S)-6-(1-benzyl-3,4,5-trimethylimidazol-3-ium-2-yl)sulfanyl-5-oxo-2-[[(2S)-3-phenyl-2-(phenylmethoxycarbonylamino)propanoyl]amino]hexanoic acid;bromide NA 200000 NA NA NA NA TTD
F13A1 (2S)-6-(1-benzyl-3,4,5-trimethylimidazol-3-ium-2-yl)sulfanyl-5-oxo-2-[[2-(phenylmethoxycarbonylamino)acetyl]amino]hexanoic acid;bromide NA 200000 NA NA NA NA TTD
F13A1 [(5S)-5-carboxy-2-oxo-5-[[2-(phenylmethoxycarbonylamino)acetyl]amino]pentyl]-diethylsulfanium;bromide NA 200000 NA NA NA NA TTD
F2 3-(6-Carbamimidoyl-benzofuran-2-yl)-2-[4-((S)-pyrrolidin-3-yloxy)-phenyl]-propionic acid NA 1000000 NA NA NA NA TTD
F2 [5-[4-[(4-Carbamimidoylphenyl)methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-(2-piperidin-4-ylethylcarbamoyl)piperazine-1-carboxylate 111000 NA NA NA NA NA TTD
F2 (S)-2-[(S)-2-((S)-2-Amino-3-phenyl-propionylamino)-4-methyl-pentanoylamino]-3-phenyl-propionic acid methyl ester NA 333000 NA NA NA NA TTD
F2 (S)-2-{(S)-2-[(S)-2-(6-Guanidino-hexanoylamino)-3-phenyl-propionylamino]-4-methyl-pentanoylamino}-3-phenyl-propionic acid methyl ester NA 200000 NA NA NA NA TTD
F2 3-(5-Carbamimidoyl-benzofuran-2-yl)-2-[4-((S)-pyrrolidin-3-yloxy)-phenyl]-propionic acid NA 230000 NA NA NA NA TTD
F2 3-(6-Carbamimidoyl-benzofuran-2-yl)-2-{4-[(S)-1-(1-imino-ethyl)-pyrrolidin-3-yloxy]-phenyl}-propionic acid NA 400000 NA NA NA NA TTD
F2 2-Acetylamino-N-[(4-carbamimidoyl-benzylcarbamoyl)-methyl]-3-hydroxy-propionamide 1000000 NA NA NA NA NA TTD
F2 H-Cys(1)-Pro-Ala-Tyr-Ser-Arg-Tyr-Leu-Asp-Cys(1)-OH 1000000 NA NA NA NA NA TTD
F2 (S)-2-{(S)-2-[(S)-2-(5-Guanidino-pentanoylamino)-3-phenyl-propionylamino]-4-methyl-pentanoylamino}-3-phenyl-propionic acid methyl ester NA 154000 NA NA NA NA TTD
F2 4-Phenyl-1-{(S)-2-[(R)-2-(thiazole-2-carbonyl)-pyrrolidine-1-carbonyl]-pyrrolidin-1-yl}-butan-1-one NA 1000000 NA NA NA NA TTD
F2 (S)-2-{(S)-2-[(S)-2-(7-Amino-heptanoylamino)-3-phenyl-propionylamino]-4-methyl-pentanoylamino}-3-phenyl-propionic acid methyl ester NA 330000 NA NA NA NA TTD
F2 3-(7-Carbamimidoyl-naphthalen-2-yl)-2-[4-((S)-pyrrolidin-3-yloxy)-phenyl]-propionic acid ethyl ester NA 600000 NA NA NA NA TTD
F2 {(R)-1-[2-(4-carbamimidoyl-benzylcarbamoyl)-indan-2-ylcarbamoyl]-2-methyl-propylamino}-acetic acid NA 300000 NA NA NA NA TTD
F2 (S)-2-{(S)-2-[(S)-2-(4-Amino-butyrylamino)-3-phenyl-propionylamino]-4-methyl-pentanoylamino}-3-phenyl-propionic acid methyl ester NA 300000 NA NA NA NA TTD
F2 [5-[4-[(4-Carbamimidoylphenyl)methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-(4-piperidin-4-ylbutanoyl)piperazine-1-carboxylate 102000 NA NA NA NA NA TTD