| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| F2 |
[Benzyloxycarbonylamino-(4-guanidino-phenyl)-methyl]-phosphonic acid diphenyl ester trifluoro-acetic acid salt |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
N-[(2R)-2-[2-[(4-carbamimidoylphenyl)methylamino]-2-oxoethyl]-3-oxomorpholin-4-yl]benzamide |
NA |
106000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
4-Nitrobenzamidine |
3162277.66 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
2-{[(1R)-1-[(2-{[(4-carbamimidoylphenyl)methyl]carbamoyl}-2,3-dihydro-1H-inden-2-yl)carbamoyl]propyl]amino}acetic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
{(R)-1-[2-(4-carbamimidoyl-benzylcarbamoyl)-indan-2-ylcarbamoyl]-2,2-dimethyl-propylamino}-acetic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
{1-[2-(4-Carbamimidoyl-benzylcarbamoyl)-indan-2-ylcarbamoyl]-1-methyl-ethylamino}-acetic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
{(R)-1-[6-(4-carbamimidoyl-benzylcarbamoyl)-6,7-dihydro-5H-[1]pyrindin-6-ylcarbamoyl]-2-methyl-propylamino}-acetic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
{(R)-1-[2-(4-carbamimidoyl-benzylcarbamoyl)-2,3-dihydro-1H-cyclopenta[b]naphthalen-2-ylcarbamoyl]-2-methyl-propylamino}-acetic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
{(R)-1-[2-(4-carbamimidoyl-benzylcarbamoyl)-2,3-dihydro-1H-phenalen-2-ylcarbamoyl]-2-methyl-propylamino}-acetic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
2-[[(2R)-1-[[9-[(4-carbamimidoylphenyl)methylcarbamoyl]-9-tricyclo[9.4.0.02,7]pentadeca-1(15),2,4,6,11,13-hexaenyl]amino]-3-methyl-1-oxobutan-2-yl]amino]acetic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
Sodium;[2-[[6-methoxy-3-[(2-methylpropan-2-yl)oxycarbonyl]-1-benzofuran-5-yl]oxymethyl]-1,3-benzothiazol-6-yl] sulfate |
NA |
146000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
Sodium;[2-[(2-methyl-1,3-benzothiazol-6-yl)oxymethyl]-1,3-benzothiazol-6-yl] sulfate |
NA |
327000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
sodium;[2-[(2-benzyl-3-ethoxycarbonyl-6-methoxy-1-benzofuran-5-yl)oxymethyl]-3-ethoxycarbonyl-1H-indol-5-yl] sulfate |
NA |
327000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
sodium;[3-ethoxycarbonyl-2-[(3-ethoxycarbonyl-2-methyl-1H-indol-5-yl)oxymethyl]-1-[(2-methylpropan-2-yl)oxycarbonyl]indol-5-yl] sulfate |
NA |
425000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
sodium;[3-ethoxycarbonyl-2-[[3-ethoxycarbonyl-2-[(3-ethoxycarbonyl-6-methoxy-2-methyl-1-benzofuran-5-yl)oxymethyl]-6-methoxy-1-benzofuran-5-yl]oxymethyl]-1H-indol-5-yl] sulfate |
NA |
304000 |
NA |
NA |
NA |
NA |
TTD |
| F2 |
3-(Dimethylamino)benzenecarboximidamide;2,4,6-trinitrophenol |
794328.23 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-N-[(3-chlorophenyl)methyl]-1-propylpyrrolidine-2-carboxamide |
1540000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-1-butyl-N-[(3-chlorophenyl)methyl]pyrrolidine-2-carboxamide |
1240000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-N-[(3-chlorophenyl)methyl]-1-(3-methylbutyl)pyrrolidine-2-carboxamide |
580000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| F2 |
(2S)-N-[(3-chlorophenyl)methyl]-1-(4-methylpentyl)pyrrolidine-2-carboxamide |
400000 |
NA |
NA |
NA |
NA |
NA |
TTD |